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Kinase Inhibitors
Activated Factor VII (Factor VIIa)
Arginase Inhibitor
Adenosine Receptor Ligands
Autotaxin Inhibitor
Bcl-2 Protein Inhibitors/Degraders
BCL-6 Protein Inhibitors
CD73 Immune Pathway Inhibitor/Modulator
Cell Cycle Modulators
Cell Metabolism Modulators
Chemotherapy
CoREST-selective Deacetylase (CoreDAC) inhibitors
Degraders (Protein Degraders)
DNA Methyltransferase Inhibtors
DNA Repair Targeted Therapy
DNA/RNA Synthesis Inhibitor/Blocker
Endoplasmic Reticulum Stress Modulator (ERSM)
Epigenetics Resch Products
Estrogen Receptor Modulators
Gamma (γ) Secretase (GS) Inhibitors
Glucocorticoid Receptor Antagonist/Modulator
Glucokinase Activator
Glutaminase Inhibitor
G-Protein-coupled Receptor Ligands
Heat Shock Protein Research Products
Hedgehog Signaling Pathway Modulators
Hippo Pathway Signaling Inhibitor
HMG-CoA Reductase
Hormone Receptor Modulators
Hydrolase Inhibitors/Modulators
IDO1 (INDOLEAMINE 2,3-DIOXYGENASE 1) Inhibitors
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
Immune Activation Agents/Modulators
Immuno/Inflammatory Mediators
Immunoproteasome Inhibitor
Immuno-oncology Modulators
Immunosuppressants/Immunochemotherapy Agents
Isomerase Inhibitor/Modulator
Kinesin Ligand/Modulator
KRAS Pathway Inhibitors
Liver X receptor (LXR) Agonist/Modulator
Metabolic Pathway Modulators
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 4 (MCT 4) Inhibitor
MTH1 (NUDT1, Human MutT Homologue)
Neuroactive Research Products
Notch/Wnt Signaling Pathway
Nuclear Export Protein Inhibitors/Modulators
Other Enzyme Inhibitors/Modulators
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Modulators
PCNA (Proliferating Cell Nuclear Antigen)
PDE4 ( Phosphodiesterase Type 4) Inhibitor/Modulators
Phosphatase Inhibitors/Modulators
PLA2 (Phospholipase A2) Inhibitor
Polymerase Inhibitor/Modulator
PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
Reagents for Biological Assays
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SMAC Mimics and Inhibitors of IAP
Stem Cell Research Products
STING (Stimulator of Interferon Genes) Agonist
SUMO Pathway Modulator
TEAD Inhibitor
Toll-like Receptor Modulators
Ubiquitin / Proteasome System
Wnt Signaling Pathway Modulators
WRN helicase Inhibitor
YAP/TAZ Signaling Inhibitor
Zinc Finger Protein Degrader
Akt/(PKB (Protein Kinase B)
ALK (Anaplastic Lymphoma Kinase)
AMPK (AMP-Activated Protein Kinase)
ASK1 (Apoptosis Signal-regulating Kinase 1)
ATM (Ataxia Telangiectasia Mutated Kinase)
ATR (Ataxia Telangiectasia and Rad3 Related)
Aurora Kinase
Aurora A Kinase Selective
Aurora B Kinase Selective
Aurora C Kinase Selective
AXL (AXL Receptor Tyrosine Kinase)
Bcr-Abl/c-kit/PDGFR/Src
BTK (Bruton's Tyrosine Kinase)
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CDK (Cyclin-dependent Kinase)
CDK2 Selective
CDK4 Selective
CDK7 Selective
CDK9 Selective
CDK12/CDK13
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
CLK2 (CDC2-like Kinase 2)
c-Met
DDK (Dbf4-dependent kinase)
DNA-PK (DNA-Dependent Protein Kinase)
EGFR Mutants
EGFR/HER2
EphB4 (Ephrin Type-B Receptor 4) Kinase
ErbB
Erk (Extracellular signal regulated kinase)
FAK (Focal Adhesion Kinase)
FGFR (Fibroblast Growth Factor Receptor)
FGFR4 Specific
FLT3 (Fms-like Tyrosine Kinase 3)
Glucokinase
IGF-1R
JAK (Janus Kinase)
JAK1 Selective
JAK1/JAK2 Selective
JAK2 Selective
JAK3 Selective
LRRK2
MEK/MAPK
Mps1 (Monopolar Spindle 1)
mTOR
PKC (Protein Kinase C)
NIK (NF-κB-inducing kinase) Inhibitors
P21-Activated Kinases
P70S6K (Ribosomal Protein S6 Kinase)
PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
PI3K - p110 Beta (β) Specific
PI3K - p110 Delta (δ) Specific
PI3K - p110 Gamma (γ) Specific
PI3K - Pan
PI3K/mTOR
PIM
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
PLK4 (Polo-like Kinase 4) Selective
PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
VEGFR
WEE1
Factor VIIa inhibitor
Bcl-2 Family Protein Inhibitors
BCL-2 Selective Inhibitors
BCL-XL Protein Degrader
BCL-XL Selective Inhibitors
MCL-1 Selective Inhibitors
CD73 (ecto-5'-nucleotidase) Inhibitor
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CBP/β-catenin Modulators
Cell Cycle/DNA Damage
CDK Inhibitors/Modulators
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
DNA Replication Modulators/Breakers
Endoplasmic Reticulum Stress Modulator (ERSM)
G-Quadruplex Ligand
IMPDH Inhibitor
Kinesin (CENP-E) Inhibitor
KRAS-G12C Inhibitors
KRASG12C (ON) (Tri-complex) Inhibitor
KRAS-G12D Inhibitors
KRAS-PDEδ Interaction Inhibitor
KRAS-SOS1 Inhibitors
Menin-KMT2A/MLL interaction inhibitors
Mps1 (Monopolar Spindle 1)
Notch Signaling Inhibitors
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
p53-MDM2 Interaction Inhibitor
PCNA (Proliferating Cell Nuclear Antigen)
PRC2 (the catalytic subunit of polycomb repressive complex 2) >
PKMYT1 Kinase Inhibitor
SMAC Mimics and Inhibitors of IAP
Survivin
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Tubulin
Wee1
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Mutant Isocitrate Dehydrogenase-1 (IDH1) Inhibitor
Mutant Isocitrate Dehydrogenase-2 (IDH2) Inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
Chemotherapy Agents
ATPases (BRG1/BRM)
BET Family Protein Degraders
BET Family Protein Inhibitors
BET/Bromodomain (BDI and BDII) Selective Inhibitors
BET/BRD4 Degrader
BET/BRD9 Degrader
BET Bromodomain II (BDII) Selective Inhibitors
BET/Domain & Sub-set Selective Inhibitors
CBP/P300 Bromodomain Inhibitor
CoreDAC Inhibitors
DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
EP300/CBP HAT (Histone Acetyltransferases) Inhibitor
EZH1/2 Dual Inhibitors
EZH2 Methyltransferase Inhibitors
EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
HDAC (histone deacetylase) Inhibitors
HDAC1-Specific Inhibitors
HDAC3-Specific Inhibitors
HDAC6-Specific Inhibitors
Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-KMT2A/MLL interaction inhibitors
PRC2 (the catalytic subunit of polycomb repressive complex 2)
PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
PRMTs (Type I) Inhibitors/Modulators
Adenosine Receptor Ligands
Angiotensin II receptor (AT1)
Endothelin receptor antagonist (type A specific)
Heat Shock Proteins HSP90 Inhibitors
Hedgehog Signaling Pathway Inhibitors
HMG-CoA reductase inhibitor
Androgen receptor
Glucocorticoid Receptor
RXRs (retinoid X receptors)
Autotaxin
Caspase-1
Cathepsin K
Glycoside Hydrolase
Neprilysin (MME)
PDE4 ( phosphodiesterase type 4)
PLA2 Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH Inhibitor
Liver X receptor (LXR) Agonist/Modulator
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
STING (STIMULATOR OF INTERFERON GENES) AGONIST
Toll-like Receptor Agonist
Anti-angiogenesis
Anti-fibrosis
Anti-inflammatory
Arginase Inhibitor
Autotaxin Inhibitors
PLA2 Inhibitors
Prostanoid ligand
RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE
TGFβ Kinase Inhibitor
Adenosine 2A Receptor Antagonist
Arginase Inhibitor
CD73 (ecto-5'-nucleotidase) Inhibitor
CBP/β-catenin Modulators
CoreDAC Inhibitors
IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
Zinc Finger Protein Degrader
Immunoproteasome Inhibitor
Liver X receptor (LXR) Agonist/Modulator
mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
PI3Kγ (GAMMA) Specific Inhibitors
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SHP2 Phosphatase Inhibitor
STING (Stimulator of Interferon Genes) Agonist
SUMOylation Inhibitor
TGFβ Kinase Inhibitor
Toll-like Receptor Modulators
Topoisomerase I
Topoisomerase II
Kinesin (CENP-E) Inhibitor
G12C Mutant Inhibitors
G12D Mutant Inhibitors
KRAS-PDEδ Interaction Inhibitor
Pan-KRAS Inhibitors
SOS1 Inhibitors
Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
MTH1
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
SDAM (Serotonin-Dopamine Activity Modulator)
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
CBP/β-catenin Modulators
Gamma (γ) Secretase (GS) Inhibitors
Notch Signaling Inhibitors
CRM1 (exportin 1) Inhibitor(s)
HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
WRN Helicase Inhibitor
p53–MDM2 Interaction Inhibitor
p53 Reactivator
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
PARP (Poly (ADP-ribose) polymerase)
Stem cell research
NADD8-Activating Enzyme Inhibtor
Proteasome Inhibitor
SUMOylation Inhibitor
Ubiquitin-Activating Enzyme Inhibitor
USP1 (Ubiquitin Specific Protease 1)
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Kinase Inhibitors
Activated Factor VII (Factor VIIa)
Arginase Inhibitor
Adenosine Receptor Ligands
Autotaxin Inhibitor
Bcl-2 Protein Inhibitors/Degraders
BCL-6 Protein Inhibitors
CD73 Immune Pathway Inhibitor/Modulator
Cell Cycle Modulators
Cell Metabolism Modulators
Chemotherapy
CoREST-selective Deacetylase (CoreDAC) inhibitors
Degraders (Protein Degraders)
DNA Methyltransferase Inhibtors
DNA Repair Targeted Therapy
DNA/RNA Synthesis Inhibitor/Blocker
Endoplasmic Reticulum Stress Modulator (ERSM)
Epigenetics Resch Products
Estrogen Receptor Modulators
Gamma (γ) Secretase (GS) Inhibitors
Glucocorticoid Receptor Antagonist/Modulator
Glucokinase Activator
Glutaminase Inhibitor
G-Protein-coupled Receptor Ligands
Heat Shock Protein Research Products
Hedgehog Signaling Pathway Modulators
Hippo Pathway Signaling Inhibitor
HMG-CoA Reductase
Hormone Receptor Modulators
Hydrolase Inhibitors/Modulators
IDO1 (INDOLEAMINE 2,3-DIOXYGENASE 1) Inhibitors
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
Immune Activation Agents/Modulators
Immuno/Inflammatory Mediators
Immunoproteasome Inhibitor
Immuno-oncology Modulators
Immunosuppressants/Immunochemotherapy Agents
Isomerase Inhibitor/Modulator
Kinesin Ligand/Modulator
KRAS Pathway Inhibitors
Liver X receptor (LXR) Agonist/Modulator
Metabolic Pathway Modulators
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 4 (MCT 4) Inhibitor
MTH1 (NUDT1, Human MutT Homologue)
Neuroactive Research Products
Notch/Wnt Signaling Pathway
Nuclear Export Protein Inhibitors/Modulators
Other Enzyme Inhibitors/Modulators
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Modulators
PCNA (Proliferating Cell Nuclear Antigen)
PDE4 ( Phosphodiesterase Type 4) Inhibitor/Modulators
Phosphatase Inhibitors/Modulators
PLA2 (Phospholipase A2) Inhibitor
Polymerase Inhibitor/Modulator
PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
Reagents for Biological Assays
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SMAC Mimics and Inhibitors of IAP
Stem Cell Research Products
STING (Stimulator of Interferon Genes) Agonist
SUMO Pathway Modulator
TEAD Inhibitor
Toll-like Receptor Modulators
Ubiquitin / Proteasome System
Wnt Signaling Pathway Modulators
WRN helicase Inhibitor
YAP/TAZ Signaling Inhibitor
Zinc Finger Protein Degrader
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New Products (II)
New & Featured Products
Kinase Inhibitors
Akt/(PKB (Protein Kinase B)
ALK (Anaplastic Lymphoma Kinase)
AMPK (AMP-Activated Protein Kinase)
ASK1 (Apoptosis Signal-regulating Kinase 1)
ATM (Ataxia Telangiectasia Mutated Kinase)
ATR (Ataxia Telangiectasia and Rad3 Related)
Aurora Kinase
Aurora A Kinase Selective
Aurora B Kinase Selective
Aurora C Kinase Selective
AXL (AXL Receptor Tyrosine Kinase)
Bcr-Abl/c-kit/PDGFR/Src
BTK (Bruton's Tyrosine Kinase)
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CDK (Cyclin-dependent Kinase)
CDK2 Selective
CDK4 Selective
CDK7 Selective
CDK9 Selective
CDK12/CDK13
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
CLK2 (CDC2-like Kinase 2)
c-Met
DDK (Dbf4-dependent kinase)
DNA-PK (DNA-Dependent Protein Kinase)
EGFR Mutants
EGFR/HER2
EphB4 (Ephrin Type-B Receptor 4) Kinase
ErbB
Erk (Extracellular signal regulated kinase)
FAK (Focal Adhesion Kinase)
FGFR (Fibroblast Growth Factor Receptor)
FGFR4 Specific
FLT3 (Fms-like Tyrosine Kinase 3)
Glucokinase
IGF-1R
JAK (Janus Kinase)
JAK1 Selective
JAK1/JAK2 Selective
JAK2 Selective
JAK3 Selective
LRRK2
MEK/MAPK
Mps1 (Monopolar Spindle 1)
mTOR
PKC (Protein Kinase C)
NIK (NF-κB-inducing kinase) Inhibitors
P21-Activated Kinases
P70S6K (Ribosomal Protein S6 Kinase)
PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
PI3K - p110 Beta (β) Specific
PI3K - p110 Delta (δ) Specific
PI3K - p110 Gamma (γ) Specific
PI3K - Pan
PI3K/mTOR
PIM
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
PLK4 (Polo-like Kinase 4) Selective
PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
VEGFR
WEE1
Activated Factor VII (Factor VIIa)
Factor VIIa inhibitor
Arginase Inhibitor
Adenosine Receptor Ligands
Autotaxin Inhibitor
Bcl-2 Protein Inhibitors/Degraders
Bcl-2 Family Protein Inhibitors
BCL-2 Selective Inhibitors
BCL-XL Protein Degrader
BCL-XL Selective Inhibitors
MCL-1 Selective Inhibitors
BCL-6 Protein Inhibitors
CD73 Immune Pathway Inhibitor/Modulator
CD73 (ecto-5'-nucleotidase) Inhibitor
Cell Cycle Modulators
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CBP/β-catenin Modulators
Cell Cycle/DNA Damage
CDK Inhibitors/Modulators
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
DNA Replication Modulators/Breakers
Endoplasmic Reticulum Stress Modulator (ERSM)
G-Quadruplex Ligand
IMPDH Inhibitor
Kinesin (CENP-E) Inhibitor
KRAS-G12C Inhibitors
KRASG12C (ON) (Tri-complex) Inhibitor
KRAS-G12D Inhibitors
KRAS-PDEδ Interaction Inhibitor
KRAS-SOS1 Inhibitors
Menin-KMT2A/MLL interaction inhibitors
Mps1 (Monopolar Spindle 1)
Notch Signaling Inhibitors
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
p53-MDM2 Interaction Inhibitor
PCNA (Proliferating Cell Nuclear Antigen)
PRC2 (the catalytic subunit of polycomb repressive complex 2) >
PKMYT1 Kinase Inhibitor
SMAC Mimics and Inhibitors of IAP
Survivin
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Tubulin
Wee1
Cell Metabolism Modulators
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Mutant Isocitrate Dehydrogenase-1 (IDH1) Inhibitor
Mutant Isocitrate Dehydrogenase-2 (IDH2) Inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
Chemotherapy
Chemotherapy Agents
CoREST-selective Deacetylase (CoreDAC) inhibitors
Degraders (Protein Degraders)
DNA Methyltransferase Inhibtors
DNA Repair Targeted Therapy
DNA/RNA Synthesis Inhibitor/Blocker
Endoplasmic Reticulum Stress Modulator (ERSM)
Epigenetics Resch Products
ATPases (BRG1/BRM)
BET Family Protein Degraders
BET Family Protein Inhibitors
BET/Bromodomain (BDI and BDII) Selective Inhibitors
BET/BRD4 Degrader
BET/BRD9 Degrader
BET Bromodomain II (BDII) Selective Inhibitors
BET/Domain & Sub-set Selective Inhibitors
CBP/P300 Bromodomain Inhibitor
CoreDAC Inhibitors
DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
EP300/CBP HAT (Histone Acetyltransferases) Inhibitor
EZH1/2 Dual Inhibitors
EZH2 Methyltransferase Inhibitors
EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
HDAC (histone deacetylase) Inhibitors
HDAC1-Specific Inhibitors
HDAC3-Specific Inhibitors
HDAC6-Specific Inhibitors
Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-KMT2A/MLL interaction inhibitors
PRC2 (the catalytic subunit of polycomb repressive complex 2)
PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
PRMTs (Type I) Inhibitors/Modulators
Estrogen Receptor Modulators
Gamma (γ) Secretase (GS) Inhibitors
Glucocorticoid Receptor Antagonist/Modulator
Glucokinase Activator
Glutaminase Inhibitor
G-Protein-coupled Receptor Ligands
Adenosine Receptor Ligands
Angiotensin II receptor (AT1)
Endothelin receptor antagonist (type A specific)
Heat Shock Protein Research Products
Heat Shock Proteins HSP90 Inhibitors
Hedgehog Signaling Pathway Modulators
Hedgehog Signaling Pathway Inhibitors
Hippo Pathway Signaling Inhibitor
HMG-CoA Reductase
HMG-CoA reductase inhibitor
Hormone Receptor Modulators
Androgen receptor
Glucocorticoid Receptor
RXRs (retinoid X receptors)
Hydrolase Inhibitors/Modulators
Autotaxin
Caspase-1
Cathepsin K
Glycoside Hydrolase
Neprilysin (MME)
PDE4 ( phosphodiesterase type 4)
PLA2 Inhibitors
IDO1 (INDOLEAMINE 2,3-DIOXYGENASE 1) Inhibitors
IDH (Isocitrate Dehydrogenase) Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
IMPDH Inhibitor
Immune Activation Agents/Modulators
Liver X receptor (LXR) Agonist/Modulator
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
STING (STIMULATOR OF INTERFERON GENES) AGONIST
Toll-like Receptor Agonist
Immuno/Inflammatory Mediators
Anti-angiogenesis
Anti-fibrosis
Anti-inflammatory
Arginase Inhibitor
Autotaxin Inhibitors
PLA2 Inhibitors
Prostanoid ligand
RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE
TGFβ Kinase Inhibitor
Immunoproteasome Inhibitor
Immuno-oncology Modulators
Adenosine 2A Receptor Antagonist
Arginase Inhibitor
CD73 (ecto-5'-nucleotidase) Inhibitor
CBP/β-catenin Modulators
CoreDAC Inhibitors
IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
Zinc Finger Protein Degrader
Immunoproteasome Inhibitor
Liver X receptor (LXR) Agonist/Modulator
mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
PI3Kγ (GAMMA) Specific Inhibitors
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SHP2 Phosphatase Inhibitor
STING (Stimulator of Interferon Genes) Agonist
SUMOylation Inhibitor
TGFβ Kinase Inhibitor
Toll-like Receptor Modulators
Immunosuppressants/Immunochemotherapy Agents
Isomerase Inhibitor/Modulator
Topoisomerase I
Topoisomerase II
Kinesin Ligand/Modulator
Kinesin (CENP-E) Inhibitor
KRAS Pathway Inhibitors
G12C Mutant Inhibitors
G12D Mutant Inhibitors
KRAS-PDEδ Interaction Inhibitor
Pan-KRAS Inhibitors
SOS1 Inhibitors
Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Liver X receptor (LXR) Agonist/Modulator
Metabolic Pathway Modulators
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4) Inhibitor
MTH1 (NUDT1, Human MutT Homologue)
MTH1
Neuroactive Research Products
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
SDAM (Serotonin-Dopamine Activity Modulator)
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
Notch/Wnt Signaling Pathway
CBP/β-catenin Modulators
Gamma (γ) Secretase (GS) Inhibitors
Notch Signaling Inhibitors
Nuclear Export Protein Inhibitors/Modulators
CRM1 (exportin 1) Inhibitor(s)
Other Enzyme Inhibitors/Modulators
HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
WRN Helicase Inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Modulators
p53–MDM2 Interaction Inhibitor
p53 Reactivator
PCNA (Proliferating Cell Nuclear Antigen)
PDE4 ( Phosphodiesterase Type 4) Inhibitor/Modulators
Phosphatase Inhibitors/Modulators
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
PLA2 (Phospholipase A2) Inhibitor
Polymerase Inhibitor/Modulator
PARP (Poly (ADP-ribose) polymerase)
PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
Reagents for Biological Assays
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SMAC Mimics and Inhibitors of IAP
Stem Cell Research Products
Stem cell research
STING (Stimulator of Interferon Genes) Agonist
SUMO Pathway Modulator
TEAD Inhibitor
Toll-like Receptor Modulators
Ubiquitin / Proteasome System
NADD8-Activating Enzyme Inhibtor
Proteasome Inhibitor
SUMOylation Inhibitor
Ubiquitin-Activating Enzyme Inhibitor
USP1 (Ubiquitin Specific Protease 1)
Wnt Signaling Pathway Modulators
WRN helicase Inhibitor
YAP/TAZ Signaling Inhibitor
Zinc Finger Protein Degrader
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Categories
PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
FX-909
Epigenetics Resch Products
>>
BET Bromodomain II (BDII) Selective Inhibitors
ABBV-744 (ABBV744)
GSK046 (IBET-BD2)
GSK973
Cell Cycle Modulators
>>
KRAS-G12D Inhibitors
MRTX1133
Liver X receptor (LXR) Agonist/Modulator
RGX-104
Epigenetics Resch Products
>>
PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
AMG-193
GSK3326595 (EPZ015938)
JNJ-64619178 (JNJ64619178)
MRTX1719
PF-06855800 (PF06855800)
PF-06939999
TNG-462
Phosphatase Inhibitors/Modulators
>>
SHP2 Phosphatase Inhibitor
GDC-1971
IACS-13909
JAB-3068
PF-07284892 (ARRY-558)
RMC-4550 (RMC4550)
RMC-4630
SHP099
TNO155
WRN helicase Inhibitor
VVD-214
Zinc Finger Protein Degrader
CFT-7455
NVP-DKY709
Immuno-oncology Modulators
>>
Adenosine 2A Receptor Antagonist
AZD4635 (HTL-1071)
PBF-509 (Taminadenant)
G-Protein-coupled Receptor Ligands
>>
Adenosine Receptor Ligands
CGS-21680
CVT-6883
Adenosine Receptor Ligands
AZD4635 (HTL-1071)
CGS-21680
CVT-6883
PBF-509 (Taminadenant)
SCH442416
Vipadenant
Kinase Inhibitors
>>
Akt/(PKB (Protein Kinase B)
Afuresertib (GSK2110183)
AZD5363
GDC-0068
GSK690693
M2698 (MSC2363318A)
MK-2206 Dihydrochloride Salt (2xHCl SALT)
MK-2206 Monohydrochloride (1 x HCl salt)
Uprosertib (GSK2141795)
Kinase Inhibitors
>>
ALK (Anaplastic Lymphoma Kinase)
AP26113 (Brigatinib)
ASP3026
AZD3463
CEP-28122
CEP-28122 Mesylate
CEP-37440
CH5424802
LDK378 (Ceritinib)
NVP-TAE684
PF-02341066
PF-06463922 (Lorlatinib)
Kinase Inhibitors
>>
AMPK (AMP-Activated Protein Kinase)
A-769662
Hormone Receptor Modulators
>>
Androgen receptor
Enzalutamide
G-Protein-coupled Receptor Ligands
>>
Angiotensin II receptor (AT1)
Eprosartan Mesylate
Valsartan
Immuno/Inflammatory Mediators
>>
Anti-angiogenesis
Pomalidomide
Immuno/Inflammatory Mediators
>>
Anti-fibrosis
GS-4997 (Selonsertib)
Pirfenidone
Immuno/Inflammatory Mediators
>>
Anti-inflammatory
GS-4997 (Selonsertib)
HA130
PF-8380
Rofecoxib
Arginase Inhibitor
CB-1158
Numidargistat
Immuno-oncology Modulators
>>
Arginase Inhibitor
CB-1158
Numidargistat
Immuno/Inflammatory Mediators
>>
Arginase Inhibitor
CB-1158
Metabolic Pathway Modulators
>>
Arginase Inhibitor
CB-1158
Kinase Inhibitors
>>
ASK1 (Apoptosis Signal-regulating Kinase 1)
GS-4997 (Selonsertib)
Kinase Inhibitors
>>
ATM (Ataxia Telangiectasia Mutated Kinase)
AZD-0156 (AZD0156)
AZD6738 (Ceralasertib)
Epigenetics Resch Products
>>
ATPases (BRG1/BRM)
FHD-286
Kinase Inhibitors
>>
ATR (Ataxia Telangiectasia and Rad3 Related)
AZD6738 (Ceralasertib)
BAY-1895344 (Elimusertib)
M-1774
Tuvusertib
VE-822 (Berzosertib)
Kinase Inhibitors
>>
Aurora A Kinase Selective
JAB-2485
LY-3295668 (AK-01)
MK-5108
MLN8237
Kinase Inhibitors
>>
Aurora B Kinase Selective
AZD1152 (Barasertib)
AZD1152-HQPA
GSK-1070916 (NMI-900)
Kinase Inhibitors
>>
Aurora C Kinase Selective
GSK-1070916 (NMI-900)
Kinase Inhibitors
>>
Aurora Kinase
AZD1152 (Barasertib)
AZD1152-HQPA
CYC-116
GSK-1070916 (NMI-900)
JAB-2485
LY-3295668 (AK-01)
MK-5108
MLN8237
VX-680
XL-228
Hydrolase Inhibitors/Modulators
>>
Autotaxin
HA130
PF-8380
Autotaxin Inhibitor
HA130
PF-8380
Immuno/Inflammatory Mediators
>>
Autotaxin Inhibitors
HA130
PF-8380
Kinase Inhibitors
>>
AXL (AXL Receptor Tyrosine Kinase)
BPI-9016M
Gilteritinib (ASP2215)
MGCD265 (Glesatinib)
R-428 (Bemcentinib)
Bcl-2 Protein Inhibitors/Degraders
>>
Bcl-2 Family Protein Inhibitors
ABT-263 (Novitoclax)
ABT-737
AZD4320 (AZD-4320)
Obatoclax
Sonrotoclax (BGB-11417)
Bcl-2 Protein Inhibitors/Degraders
>>
BCL-2 Selective Inhibitors
ABT-199 (Venetoclax)
BCL-201 (S55746)
Sonrotoclax (BGB-11417)
BCL-6 Protein Inhibitors
OICR-12694 (JNJ-65234637)
Bcl-2 Protein Inhibitors/Degraders
>>
BCL-XL Protein Degrader
DT-2216
Bcl-2 Protein Inhibitors/Degraders
>>
BCL-XL Selective Inhibitors
A-1155463
A-1331852
DT-2216
WEHI-539
Kinase Inhibitors
>>
Bcr-Abl/c-kit/PDGFR/Src
AZD0530
Dasatinib
DCC-2036 (Rebastinib)
Imatinib (free base)
Nilotinib
Ponatinib
Epigenetics Resch Products
>>
BET Family Protein Degraders
ARV-825
CFT-8634
dBET1
Epigenetics Resch Products
>>
BET Family Protein Inhibitors
ABBV-744 (ABBV744)
AZD5153 (AZD-5153)
BMS-986158 (BMS986158)
GSK046 (IBET-BD2)
I-BET151 (GSK1210151A)
I-BET726 (GSK1324726A)
I-BET762 (Molibresib) (GSK525762)
JQ1, (+)
OTX-015 (Birabresib)
Pelabresib
Epigenetics Resch Products
>>
BET/BRD4 Degrader
ARV-825
dBET1
Epigenetics Resch Products
>>
BET/BRD9 Degrader
CFT-8634
Epigenetics Resch Products
>>
BET/Bromodomain (BDI and BDII) Selective Inhibitors
AZD5153 (AZD-5153)
BMS-986158 (BMS986158)
GSK046 (IBET-BD2)
GSK778 (iBET-BD1)
GSK973
JQ1, (+)
Pelabresib
Epigenetics Resch Products
>>
BET/Domain & Sub-set Selective Inhibitors
ABBV-744 (ABBV744)
AZD5153 (AZD-5153)
BMS-986158 (BMS986158)
GSK046 (IBET-BD2)
GSK778 (iBET-BD1)
GSK973
JQ1, (+)
Pelabresib
Kinase Inhibitors
>>
BTK (Bruton's Tyrosine Kinase)
Acalabrutinib (ACP196)
AVL-292 (Spebrutinib)
PCI-32765 (Ibrutinib)
Pirtobrutinib
RN486 (RN-486)
Kinase Inhibitors
>>
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
BAY-1816032 (BAY1816032)
Cell Cycle Modulators
>>
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
BAY-1816032 (BAY1816032)
Hydrolase Inhibitors/Modulators
>>
Caspase-1
VX-765 (Belnacasan)
Hydrolase Inhibitors/Modulators
>>
Cathepsin K
Odanacatib
Epigenetics Resch Products
>>
CBP/P300 Bromodomain Inhibitor
CCS-1477 (CCS1477)
Notch/Wnt Signaling Pathway
>>
CBP/β-catenin Modulators
C-82
E7386
E-7386
Foscenvivint (PRI-724)
ICG-001
Immuno-oncology Modulators
>>
CBP/β-catenin Modulators
E7386
E-7386
Cell Cycle Modulators
>>
CBP/β-catenin Modulators
C-82
E7386
E-7386
Foscenvivint (PRI-724)
ICG-001
CD73 Immune Pathway Inhibitor/Modulator
>>
CD73 (ecto-5'-nucleotidase) Inhibitor
AB-680
Immuno-oncology Modulators
>>
CD73 (ecto-5'-nucleotidase) Inhibitor
AB-680
Kinase Inhibitors
>>
CDC7 (Cell Division Cycle 7-related Protein Kinase)
LY-3177833 (LY3177833)
TAK-931 (Simurosertib)
Cell Cycle Modulators
>>
CDC7 (Cell Division Cycle 7-related Protein Kinase)
LY-3177833 (LY3177833)
Kinase Inhibitors
>>
CDK (Cyclin-dependent Kinase)
Abemaciclib Mesylate
AMG-925
Atirmociclib (PF-07220060)
AZD4573 (AZD-4573)
AZD8421
BAY-1251152 (BAY 1251152)
CT-7001 (Samuraciclib) ( ICEC0942)
Dinaciclib
KB-0742
LEE011 (Ribociclib)
LY2835219 (Abemaciclib) (Free Base)
Palbociclib (PD-0332991) (Free Base)
Palbociclib (PD-0332991) (HCl Salt)
Palbociclib Isethionate
PF-06873600
PF-07104091
THZ-531
Voruciclib
Cell Cycle Modulators
>>
CDK Inhibitors/Modulators
AMG-925
AZD4573 (AZD-4573)
CT-7001 (Samuraciclib) ( ICEC0942)
Dinaciclib
KB-0742
LEE011 (Ribociclib)
LY2835219 (Abemaciclib) (Free Base)
Palbociclib (PD-0332991) (Free Base)
Palbociclib (PD-0332991) (HCl Salt)
Palbociclib Isethionate
PF-06873600
PF-07104091
Voruciclib
Kinase Inhibitors
>>
CDK12/CDK13
SR-4835
THZ-531
Kinase Inhibitors
>>
CDK2 Selective
AZD8421
PF-06873600
PF-07104091
Kinase Inhibitors
>>
CDK4 Selective
Abemaciclib Mesylate
AMG-925
Atirmociclib (PF-07220060)
LEE011 (Ribociclib)
LY2835219 (Abemaciclib) (Free Base)
Palbociclib (PD-0332991) (Free Base)
Palbociclib (PD-0332991) (HCl Salt)
Palbociclib Isethionate
PF-06873600
Kinase Inhibitors
>>
CDK7 Selective
CT-7001 (Samuraciclib) ( ICEC0942)
KRLS-017
Kinase Inhibitors
>>
CDK9 Selective
AZD4573 (AZD-4573)
BAY-1251152 (BAY 1251152)
KB-0742
Voruciclib
Cell Cycle Modulators
>>
Cell Cycle/DNA Damage
AZD-0156 (AZD0156)
VE-822 (Berzosertib)
Chemotherapy
>>
Chemotherapy Agents
5-Azacitidine
CNDAC (DFP-10917, TAS-109)
Decitabine
Doxorubicin
Gemcitabine (Free Base)
Gemcitabine (HCl salt)
NUC-1031 (Acelarin)
Kinase Inhibitors
>>
CHK (Checkpoint Kinase)
ART-446
AZD7762
BBI-355
CCT-245737 (PNT-737)
LY-2606368 (Prexasertib) Dihydrochloride
LY2606368 (Prexasertib) Mesylate
SCH900776 (MK-8776)
Cell Cycle Modulators
>>
CHK (Checkpoint Kinase)
AZD7762
CCT-245737 (PNT-737)
LY-2606368 (Prexasertib) Dihydrochloride
SCH900776 (MK-8776)
Cell Cycle Modulators
>>
CLK (CDC2-like-Kinase)
CC-671
CTX-712 (Rogocekib)
Kinase Inhibitors
>>
CLK (CDC2-like-Kinase)
CTX-712 (Rogocekib)
Kinase Inhibitors
>>
CLK2 (CDC2-like Kinase 2)
CC-671
Kinase Inhibitors
>>
c-Met
Altiratinib (DCC-2701)
AMG-337
ARQ-197
BMS-777607
BPI-9016M
Capmatinib (INCB-28060)
Foretinib
MGCD265 (Glesatinib)
MGCD516 (Sitravatinib)
PF-02341066
PF-04217903
Volitinib (AZD6094, Savolitinib)
XL184 (Cabozantinib) (free base)
Epigenetics Resch Products
>>
CoreDAC Inhibitors
TNG-260
Immuno-oncology Modulators
>>
CoreDAC Inhibitors
TNG-260
CoREST-selective Deacetylase (CoreDAC) inhibitors
TNG-260
Nuclear Export Protein Inhibitors/Modulators
>>
CRM1 (exportin 1) Inhibitor(s)
KPT-330 (Selinexor)
Kinase Inhibitors
>>
DDK (Dbf4-dependent kinase)
LY-3177833 (LY3177833)
TAK-931 (Simurosertib)
Degraders (Protein Degraders)
ACBI1
ARV-825
CFT-1946
CFT-7455
CFT-8634
dBET1
DT-2216
NVP-DKY709
DNA Methyltransferase Inhibtors
5-Azacitidine
Decitabine
GSK-3484862 (GSKMI-714)
GSK3685032
DNA Repair Targeted Therapy
AZD7648
Cell Cycle Modulators
>>
DNA Replication Modulators/Breakers
CNDAC (DFP-10917, TAS-109)
Gemcitabine (Free Base)
Gemcitabine (HCl salt)
DNA/RNA Synthesis Inhibitor/Blocker
CNDAC (DFP-10917, TAS-109)
Gemcitabine (Free Base)
Gemcitabine (HCl salt)
NUC-1031 (Acelarin)
Kinase Inhibitors
>>
DNA-PK (DNA-Dependent Protein Kinase)
AZD7648
Epigenetics Resch Products
>>
DNMT1 (DNA Methyltransferase 1) inhibitor
5-Azacitidine
Decitabine
GSK-3484862 (GSKMI-714)
GSK3685032
Epigenetics Resch Products
>>
DOT1L Methyltransferase Inhibitor
EPZ-5676 (Pinometostat)
Kinase Inhibitors
>>
EGFR Mutants
AZ5104
AZD9291 (Osimertinib)
CO-1686 (Rociletinib)
Lazertinib
Olmutinib (BI 1482694, HM71224)
ORIC-114 | Enozertinib
TAK-788 (Mobocertinib)
TAS2940 (TAS-2940)
TAS6417
WZ4002
Kinase Inhibitors
>>
EGFR/HER2
BIBW-2992 (Afatinib)
Erlotinib
Gefitinib
Lapatinib (free base)
Lazertinib
ORIC-114 | Enozertinib
TAS2940 (TAS-2940)
Tucatinib
Endoplasmic Reticulum Stress Modulator (ERSM)
M-3913
Cell Cycle Modulators
>>
Endoplasmic Reticulum Stress Modulator (ERSM)
M-3913
G-Protein-coupled Receptor Ligands
>>
Endothelin receptor antagonist (type A specific)
Epigenetics Resch Products
>>
EP300/CBP HAT (Histone Acetyltransferases) Inhibitor
DS-9300
Kinase Inhibitors
>>
EphB4 (Ephrin Type-B Receptor 4) Kinase
NVP-BHG712 (BHG-712)
Kinase Inhibitors
>>
ErbB
BMS-599626
Dacomitinib
Kinase Inhibitors
>>
Erk (Extracellular signal regulated kinase)
GDC-0994 (Ravoxertinib, RG7842)
Hypothemycin
LY-3214996 (Temuterkib)
SCH772984
SCH900353 (MK-8353)
Ulixertinib (BVD-523, VRT752271)
VX-11e
Estrogen Receptor Modulators
ErSO
ErSO-DFP
Epigenetics Resch Products
>>
EZH1/2 Dual Inhibitors
Valemetostat (DS-3201) (DS-3201b)
Epigenetics Resch Products
>>
EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
EPZ011989
EPZ-6438 (Tazemetostat)
GSK126
PF-06821497 (PF06821497)
Epigenetics Resch Products
>>
EZH2 Methyltransferase Inhibitors
EPZ005687
EPZ011989
EPZ-6438 (Tazemetostat)
GSK126
PF-06821497 (PF06821497)
Valemetostat (DS-3201) (DS-3201b)
Activated Factor VII (Factor VIIa)
>>
Factor VIIa inhibitor
PCI-27483
Kinase Inhibitors
>>
FAK (Focal Adhesion Kinase)
CEP-37440
Defactinib (VS-6063, PF-04554878)
GSK2256098
TAE226 (NVP-TAE226)
VS-4718 (PND-1186)
Kinase Inhibitors
>>
FGFR (Fibroblast Growth Factor Receptor)
AZD4547
Erdafitinib (JNJ-42756493)
NVP-BGJ398 (Infigratinib)
Kinase Inhibitors
>>
FGFR4 Specific
Kinase Inhibitors
>>
FLT3 (Fms-like Tyrosine Kinase 3)
AC220 (Quizartinib)
Crenolanib
Gilteritinib (ASP2215)
KRAS Pathway Inhibitors
>>
G12C Mutant Inhibitors
AMG-510
ARS-1620
GDC-6036
MRTX1257 (MRTX-1257)
MRTX849
KRAS Pathway Inhibitors
>>
G12D Mutant Inhibitors
MRTX1133
RMC-9805 | Zoldonrasib
Gamma (γ) Secretase (GS) Inhibitors
Nirogacestat (PF-03084014)
Notch/Wnt Signaling Pathway
>>
Gamma (γ) Secretase (GS) Inhibitors
Hormone Receptor Modulators
>>
Glucocorticoid Receptor
CORT125134 (Relacorilant) ( CORT-125134)
Glucocorticoid Receptor Antagonist/Modulator
CORT125134 (Relacorilant) ( CORT-125134)
Kinase Inhibitors
>>
Glucokinase
MK-0941 Mesylate
Glucokinase Activator
MK-0941 Mesylate
Metabolic Pathway Modulators
>>
Glutaminase Inhibitor
CB-839 (Telaglenastat)
Glutaminase Inhibitor
CB-839 (Telaglenastat)
Hydrolase Inhibitors/Modulators
>>
Glycoside Hydrolase
ASN90
Cell Cycle Modulators
>>
G-Quadruplex Ligand
Pyridostatin
Other Enzyme Inhibitors/Modulators
>>
HCV Protease Inhibitor
VX-950
Epigenetics Resch Products
>>
HDAC (histone deacetylase) Inhibitors
Belinostat
CUDC-101
LBH-589
MGCD0103
MS-275
Romidepsin
SR-4370
Vorinostat
Epigenetics Resch Products
>>
HDAC1-Specific Inhibitors
TNG-260
Epigenetics Resch Products
>>
HDAC3-Specific Inhibitors
SR-4370
Epigenetics Resch Products
>>
HDAC6-Specific Inhibitors
Compound 7 (HCl salt)
Tubacin
Tubastatin A
WT161 (WT-161)
Heat Shock Protein Research Products
>>
Heat Shock Proteins HSP90 Inhibitors
CUDC-305 (DEBIO-0932)
NVP-AUY922
Hedgehog Signaling Pathway Modulators
>>
Hedgehog Signaling Pathway Inhibitors
GDC-0449 (Vismodegib)
NVP-LDE225 Diphosphate salt (Erismodegib, Sonidegib)
Hippo Pathway Signaling Inhibitor
GNE-7883
IAG933
IK-930
NVP-IAG933
VT-107
Other Enzyme Inhibitors/Modulators
>>
HIV-1 integrase Inhibitor
Raltegravir
HMG-CoA Reductase
>>
HMG-CoA reductase inhibitor
Atorvastatin Calcium
Metabolic Pathway Modulators
>>
IDH (Isocitrate Dehydrogenase) Inhibitors
AG-120 (Ivosidenib)
AG-221 (Enasidenib)
BAY-1436032
Immuno-oncology Modulators
>>
IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
Epacadostat
LY-3381916
PF-06840003 (EOS-200271)
IDO1 (INDOLEAMINE 2,3-DIOXYGENASE 1) Inhibitors
Epacadostat
LY-3381916
PF-06840003 (EOS-200271)
Kinase Inhibitors
>>
IGF-1R
BMS-754807
GSK1904529A
OSI-906 (Linsitinib)
TAE226 (NVP-TAE226)
XL-228
Immunoproteasome Inhibitor
M-3258
Immuno-oncology Modulators
>>
Immunoproteasome Inhibitor
M-3258
Immunosuppressants/Immunochemotherapy Agents
Darovasertib (NVP-LXS196)
Everolimus
PD-1 Inhibitor 16 (Aurigene Compound 16)
Rapamycin (Sirolimus)
Metabolic Pathway Modulators
>>
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
AVN944
Cell Cycle Modulators
>>
IMPDH Inhibitor
AVN944
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
>>
IMPDH Inhibitor
AVN944
Kinase Inhibitors
>>
JAK (Janus Kinase)
ASN-002 (Gusacitinib)
AZD1480
AZD-4205 (AZD4205)
BMS-911543
Cerdulatinib
CYT-387 (Momelotinib)
Decernotinib (VX-509)
GLPG-0634 (Filgotinib)
INCB018424 (Ruxolitinib)
Ruxolitinib Phosphate
TG101348 (Fedratinib, SAR302503)
Upadacitinib (ABT-494)
Kinase Inhibitors
>>
JAK1 Selective
AZD-4205 (AZD4205)
GLPG-0634 (Filgotinib)
Upadacitinib (ABT-494)
Kinase Inhibitors
>>
JAK1/JAK2 Selective
AZD1480
CYT-387 (Momelotinib)
INCB018424 (Ruxolitinib)
Ruxolitinib Phosphate
Kinase Inhibitors
>>
JAK2 Selective
BMS-911543
TG101348 (Fedratinib, SAR302503)
Kinase Inhibitors
>>
JAK3 Selective
Decernotinib (VX-509)
Kinesin Ligand/Modulator
>>
Kinesin (CENP-E) Inhibitor
GSK923295
Cell Cycle Modulators
>>
Kinesin (CENP-E) Inhibitor
GSK923295
Cell Cycle Modulators
>>
KRASG12C (ON) (Tri-complex) Inhibitor
RMC-6291 | Elironrasib
Cell Cycle Modulators
>>
KRAS-G12C Inhibitors
AMG-510
ARS-1620
GDC-6036
MRTX1257 (MRTX-1257)
MRTX849
Cell Cycle Modulators
>>
KRAS-PDEδ Interaction Inhibitor
Deltarasin HCl salt
KRAS Pathway Inhibitors
>>
KRAS-PDEδ Interaction Inhibitor
Deltarasin HCl salt
Cell Cycle Modulators
>>
KRAS-SOS1 Inhibitors
BAY-293
BI-3406
MRTX0902
Immune Activation Agents/Modulators
>>
Liver X receptor (LXR) Agonist/Modulator
Immuno-oncology Modulators
>>
Liver X receptor (LXR) Agonist/Modulator
RGX-104
Kinase Inhibitors
>>
LRRK2
GNE-7915
Epigenetics Resch Products
>>
Lysine specific demethylase 1 (LSD1) Inhibitor
GSK2879552
Metabolic Pathway Modulators
>>
MAT2A Inhibitor
Bcl-2 Protein Inhibitors/Degraders
>>
MCL-1 Selective Inhibitors
A-1210477
ABBV-467
AMG-176 (Tapotoclax)
AZD5991 (AZD-5991)
MIK665
S63845 (S-63845)
S64315
Kinase Inhibitors
>>
MEK/MAPK
Arry-162 (Binimetinib, MEK162)
AS-703026 (Pimasertib)
AZD6244 (Selumetinib)
AZD8330
GDC-0973 (Cobimetinib)
GSK1120212 (Trametinib)
PD-0325901
RDEA119 (Refametinib)
VX-702
Epigenetics Resch Products
>>
Menin-KMT2A/MLL interaction inhibitors
Enzomenib | DSP-5336
JNJ- 75276617 (Bleximenib)
Ziftomenib (KO-539)
Cell Cycle Modulators
>>
Menin-KMT2A/MLL interaction inhibitors
Enzomenib | DSP-5336
JNJ- 75276617 (Bleximenib)
Ziftomenib (KO-539)
Metabolic Pathway Modulators
>>
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
AZD3965
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
>>
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
AZD3965
Cell Metabolism Modulators
>>
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
AZD3965
Metabolic Pathway Modulators
>>
Monocarboxylate Transporter 4 (MCT 4)
AZD0095
Monocarboxylate Transporter 4 (MCT 4) Inhibitor
AZD0095
Kinase Inhibitors
>>
Mps1 (Monopolar Spindle 1)
Cell Cycle Modulators
>>
Mps1 (Monopolar Spindle 1)
CC-671
MTH1 (NUDT1, Human MutT Homologue)
>>
MTH1
Crizotinib, S-enantiomer
Kinase Inhibitors
>>
mTOR
AZD2014 (Vistusertib)
AZD8055
Everolimus
OSI-027
Pp242
Rapamycin (Sirolimus)
Sapanisertib (TAK-228) (MLN0128)
TORIN 2
Immuno-oncology Modulators
>>
mTOR inhibitors
Everolimus
Rapamycin (Sirolimus)
Cell Metabolism Modulators
>>
Mutant Isocitrate Dehydrogenase-1 (IDH1) Inhibitor
AG-120 (Ivosidenib)
BAY-1436032
Cell Metabolism Modulators
>>
Mutant Isocitrate Dehydrogenase-2 (IDH2) Inhibitor
AG-221 (Enasidenib)
IDH (Isocitrate Dehydrogenase) Inhibitors
>>
Mutant-IDH1 Inhibitor
AG-120 (Ivosidenib)
BAY-1436032
IDH (Isocitrate Dehydrogenase) Inhibitors
>>
Mutant-IDH2 Inhibitor
AG-221 (Enasidenib)
Ubiquitin / Proteasome System
>>
NADD8-Activating Enzyme Inhibtor
MLN4924 (Pevonedistat)
Hydrolase Inhibitors/Modulators
>>
Neprilysin (MME)
AHU-377 (Sacubitril)
Neuroactive Research Products
>>
Neuroactive/BBB Penetrant
Altiratinib (DCC-2701)
AP26113 (Brigatinib)
ASN90
CUDC-305 (DEBIO-0932)
FRAX486
GNE-7915
J-147
Lazertinib
M2698 (MSC2363318A)
NVP-LDE225 Diphosphate salt (Erismodegib, Sonidegib)
ORIC-114 | Enozertinib
PBF-509 (Taminadenant)
PF-06463922 (Lorlatinib)
PF-06840003 (EOS-200271)
TAS2940 (TAS-2940)
New & Featured Products
AB-680
ADU-S100 (MIW815)
AMG-176 (Tapotoclax)
AZD5991 (AZD-5991)
CB-1158
CFT-8634
cGAMP
CT-7001 (Samuraciclib) ( ICEC0942)
DT-2216
E-7766
GDC-6036
GSK3685032
KB-0742
LHC-165
LXH254 (Naporafenib)
M-3258
MRTX1257 (MRTX-1257)
MRTX1719
NVP-HDM201 (Siremadlin) (HDM-201)
PF-06821497 (PF06821497)
PF-06873600
PF-06939999
PF-07104091
S64315
New Products (II)
ABBV-467
ASTX295 | ASTX-295
BI-907828 (Brigimadlin)
CFT-1946
Enzomenib | DSP-5336
JAB-2485
MK-2118
OICR-12694 (JNJ-65234637)
Rezatapopt
RMC-6236
RMC-6291 | Elironrasib
RMC-7977
RMC-9805 | Zoldonrasib
SNX281
Sonrotoclax (BGB-11417)
VVD-214
Kinase Inhibitors
>>
NIK (NF-κB-inducing kinase) Inhibitors
NIK SMI1
Cell Cycle Modulators
>>
Notch Signaling Inhibitors
CB-103
Notch/Wnt Signaling Pathway
>>
Notch Signaling Inhibitors
CB-103
Neuroactive Research Products
>>
Orexin Receptor Antagonists
MK-3697
Other Enzyme Inhibitors/Modulators
>>
Oxidoreductase Inhibitor
Dutasteride
Metabolic Pathway Modulators
>>
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
IACS-010759 (IACS-10759)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
IACS-010759 (IACS-10759)
Cell Cycle Modulators
>>
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
IACS-010759 (IACS-10759)
Cell Metabolism Modulators
>>
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
IACS-010759 (IACS-10759)
Kinase Inhibitors
>>
P21-Activated Kinases
FRAX486
PF-03758309
p53–MDM2 Modulators
>>
p53 Reactivator
Rezatapopt
Cell Cycle Modulators
>>
p53-MDM2 Interaction Inhibitor
AMG-232
ASTX295 | ASTX-295
BI-907828 (Brigimadlin)
DS-3032 (Milademetan) (DS-3032b)
NVP-CGM097 (Free Base)
NVP-CGM097 Hydrochloride (HCl salt)
NVP-HDM201 (Siremadlin) (HDM-201)
RG7388 (Idasanutlin)
p53–MDM2 Modulators
>>
p53–MDM2 Interaction Inhibitor
AMG-232
ASTX295 | ASTX-295
BI-907828 (Brigimadlin)
DS-3032 (Milademetan) (DS-3032b)
NVP-CGM097 (Free Base)
NVP-CGM097 Hydrochloride (HCl salt)
NVP-HDM201 (Siremadlin) (HDM-201)
RG7388 (Idasanutlin)
Kinase Inhibitors
>>
P70S6K (Ribosomal Protein S6 Kinase)
M2698 (MSC2363318A)
KRAS Pathway Inhibitors
>>
Pan-KRAS Inhibitors
BI-2865
Daraxonrasib | CAS No 2765081-21-6
RMC-6236
RMC-7977
RMC-7977 | Bulk Discount |
Polymerase Inhibitor/Modulator
>>
PARP (Poly (ADP-ribose) polymerase)
ABT-888 (Veliparib)
AG014699 (Rucaparib)
AZD2281 (Olaparib)
BMN-673 (Talazoparib) (MDV-3800) (LT 00673)
BSI-201
MK-4827 (Niraparib)
Cell Cycle Modulators
>>
PCNA (Proliferating Cell Nuclear Antigen)
PCNA (Proliferating Cell Nuclear Antigen)
PD-1/PD-L1 Checkpoint Inhibitors
PD-1 Inhibitor 16 (Aurigene Compound 16)
Immuno-oncology Modulators
>>
PD-1/PD-L1 CHECKPOINT INHIBITORS
PD-1 Inhibitor 16 (Aurigene Compound 16)
Hydrolase Inhibitors/Modulators
>>
PDE4 ( phosphodiesterase type 4)
AN2728 (Crisaborole)
Apremilast
PDE4 ( Phosphodiesterase Type 4) Inhibitor/Modulators
AN2728 (Crisaborole)
Apremilast
Kinase Inhibitors
>>
PDGFR
Crenolanib
MGCD516 (Sitravatinib)
Sunitinib
Kinase Inhibitors
>>
PDK1
GSK2334470
Kinase Inhibitors
>>
PI3K - p110 Alpha (α) Specific
BAY-1082439
BYL719 (Alpelisib)
PIK-75
Serabelisib (MLN1117, INK1117, TAK-117)
Kinase Inhibitors
>>
PI3K - p110 Beta (β) Specific
AZD8186
BAY-1082439
GSK2636771
TGX-221
Kinase Inhibitors
>>
PI3K - p110 Delta (δ) Specific
CAL-101
GS-9901
IC-87114
IPI-145
Kinase Inhibitors
>>
PI3K - p110 Gamma (γ) Specific
AS-605240
AZD3458 (AZD-3458)
IPI-549
TG100-115
Kinase Inhibitors
>>
PI3K - Pan
AMG-511
GDC-0032 (Taselisib)
GDC-0941 (free base)
LY294002
NVP-BKM120 (Buparlisib)
XL-147
Kinase Inhibitors
>>
PI3K/mTOR
GDC-0980
GSK2126458 (Omipalisib)
NVP-BEZ235
PF-04691502
XL765 (Voxtalisib, SAR245409)
Immuno-oncology Modulators
>>
PI3Kγ (GAMMA) Specific Inhibitors
AZD3458 (AZD-3458)
IPI-549
Kinase Inhibitors
>>
PIM
Kinase Inhibitors
>>
PKC (Protein Kinase C)
Darovasertib (NVP-LXS196)
Kinase Inhibitors
>>
PKMYT1
RP-6306 (Lunresertib)
Cell Cycle Modulators
>>
PKMYT1 Kinase Inhibitor
RP-6306 (Lunresertib)
PLA2 (Phospholipase A2) Inhibitor
Darapladib (SB-480848)
Varespladib (LY315920)
Varespladib Methyl (LY333013)
Varespladib Sodium (LY315920 Sodium Salt)
Immuno/Inflammatory Mediators
>>
PLA2 Inhibitors
Darapladib (SB-480848)
Varespladib (LY315920)
Varespladib Methyl (LY333013)
Varespladib Sodium (LY315920 Sodium Salt)
Hydrolase Inhibitors/Modulators
>>
PLA2 Inhibitors
Darapladib (SB-480848)
Varespladib (LY315920)
Varespladib Methyl (LY333013)
Varespladib Sodium (LY315920 Sodium Salt)
Kinase Inhibitors
>>
PLK (Polo-like kinase)
BI 2536
BI 6727 (Volasertib)
GSK461364
NMS1286937 (NMS-P937)
Kinase Inhibitors
>>
PLK1 (Polo-like Kinase 1) Selective
GSK461364
NMS1286937 (NMS-P937)
Kinase Inhibitors
>>
PLK4 (Polo-like Kinase 4) Selective
Other Enzyme Inhibitors/Modulators
>>
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
RX-5902 (Supinoxin)
Epigenetics Resch Products
>>
PRC2 (the catalytic subunit of polycomb repressive complex 2)
EED-226 (EED226)
Cell Cycle Modulators
>>
PRC2 (the catalytic subunit of polycomb repressive complex 2) >
EED-226 (EED226)
Epigenetics Resch Products
>>
PRMTs (Type I) Inhibitors/Modulators
GSK3368715 (EPZ019997)
Immuno/Inflammatory Mediators
>>
Prostanoid ligand
AP-761
AP-768
Laropiprant
Ramatroban
TM30089
Ubiquitin / Proteasome System
>>
Proteasome Inhibitor
Bortezomib
Carfilzomib
MLN9708
Oprozomib
Kinase Inhibitors
>>
PTEF-b/CDK9
BAY-1251152 (BAY 1251152)
Phosphatase Inhibitors/Modulators
>>
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
ABBV-CLS-484
Osunprotafib
Immuno-oncology Modulators
>>
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
ABBV-CLS-484
Osunprotafib
Kinase Inhibitors
>>
RAF (Rapidly Accelerated Fibrosarcoma)
Belvarafenib (GDC-5573) (HM95573)
BGB-283 (Lifirafenib)
CCT196969
CFT-1946
Dabrafenib (free base)
Dabrafenib Mesylate
LGX818 (Encorafenib)
LXH254 (Naporafenib)
MLN-2480 (Tovorafenib)
PF-07799933 (Claturafenib)
PLX4032
PLX4720
Regorafenib
Sorafenib (free base)
TAK-632
Reagents for Biological Assays
D-Luciferin Potassium salt
Kinase Inhibitors
>>
RET (Rearranged During Transfection) Kinase
BLU-667 (Pralsetinib)
LOXO-292 (Selpercatinib)
MGCD516 (Sitravatinib)
Kinase Inhibitors
>>
RIP1 (Receptor Interacting Protein 1) Kinase
GSK2982772
Immuno/Inflammatory Mediators
>>
RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE
GSK2982772
Kinase Inhibitors
>>
ROCK (Rho-Associated Protein Kinase)
RKI-1447
Y-27632 Dihydrochloride
Immune Activation Agents/Modulators
>>
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
LYC-55716 (Cintirorgon) (LYC55716)
Immuno-oncology Modulators
>>
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
LYC-55716 (Cintirorgon) (LYC55716)
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
LYC-55716 (Cintirorgon) (LYC55716)
Kinase Inhibitors
>>
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Entrectinib
Hormone Receptor Modulators
>>
RXRs (retinoid X receptors)
Bexarotene
Neuroactive Research Products
>>
SDAM (Serotonin-Dopamine Activity Modulator)
Brexpiprazole (OPC-34712)
Immuno-oncology Modulators
>>
SHP2 Phosphatase Inhibitor
GDC-1971
IACS-13909
JAB-3068
PF-07284892 (ARRY-558)
RMC-4550 (RMC4550)
RMC-4630
SHP099
TNO155
SMAC Mimics and Inhibitors of IAP
AZD5582
Birinapant
LCL-161
Cell Cycle Modulators
>>
SMAC Mimics and Inhibitors of IAP
AZD5582
Birinapant
LCL-161
KRAS Pathway Inhibitors
>>
SOS1 Inhibitors
BAY-293
BI-3406
MRTX0902
Stem Cell Research Products
>>
Stem cell research
StemRegenin 1
Immune Activation Agents/Modulators
>>
STING (STIMULATOR OF INTERFERON GENES) AGONIST
2′,3′-cGAMP
ADU-S100 (MIW815)
cGAMP
E-7766
MSA-2
STING (Stimulator of Interferon Genes) Agonist
2′,3′-cGAMP
ADU-S100 (MIW815)
cGAMP
E-7766
MK-2118
MSA-2
SNX281
Immuno-oncology Modulators
>>
STING (Stimulator of Interferon Genes) Agonist
2′,3′-cGAMP
ADU-S100 (MIW815)
cGAMP
E-7766
MK-2118
MSA-2
SNX281
SUMO Pathway Modulator
TAK-981
Ubiquitin / Proteasome System
>>
SUMOylation Inhibitor
TAK-981
Immuno-oncology Modulators
>>
SUMOylation Inhibitor
TAK-981
Cell Cycle Modulators
>>
Survivin
YM155
Kinase Inhibitors
>>
Syk (Spleen Tyrosine Kinase)
ASN-002 (Gusacitinib)
Cerdulatinib
GS-9973 (Entospletinib)
TEAD Inhibitor
GNE-7883
IAG933
IK-930
NVP-IAG933
VT-107
Kinase Inhibitors
>>
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
LY-3200882 (LY3200882)
Immuno-oncology Modulators
>>
TGFβ Kinase Inhibitor
LY-3200882 (LY3200882)
Immuno/Inflammatory Mediators
>>
TGFβ Kinase Inhibitor
LY-3200882 (LY3200882)
Other Enzyme Inhibitors/Modulators
>>
Thymidylate synthase inhibitor
Immune Activation Agents/Modulators
>>
Toll-like Receptor Agonist
LHC-165
Immuno-oncology Modulators
>>
Toll-like Receptor Modulators
GS-9688 (Selgantolimod)
LHC-165
TAK-242 (Resatorvid)
Toll-like Receptor Modulators
GS-9688 (Selgantolimod)
LHC-165
TAK-242 (Resatorvid)
Kinase Inhibitors
>>
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
OTS-964
Isomerase Inhibitor/Modulator
>>
Topoisomerase I
SN-38
Topotecan
Isomerase Inhibitor/Modulator
>>
Topoisomerase II
Doxorubicin
Etoposide phosphate
KRAS Pathway Inhibitors
>>
Tri-complex KRAS inhibitors
RMC-6236
RMC-6291 | Elironrasib
RMC-7977
RMC-9805 | Zoldonrasib
KRAS Pathway Inhibitors
>>
Tri-complex KRASG12C (ON) Inhibitor
RMC-6291 | Elironrasib
Kinase Inhibitors
>>
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
Entrectinib
LOXO-101 (Larotrectinib)
LOXO-195 (Selitrectinib)
Neuroactive Research Products
>>
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
LOXO-101 (Larotrectinib)
LOXO-195 (Selitrectinib)
Kinase Inhibitors
>>
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Cell Cycle Modulators
>>
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Cell Cycle Modulators
>>
Tubulin
Docetaxel
Paclitaxel
Ubiquitin / Proteasome System
>>
Ubiquitin-Activating Enzyme Inhibitor
MLN7243 (TAK-243, AOB 87172)
Ubiquitin / Proteasome System
>>
USP1 (Ubiquitin Specific Protease 1)
KSQ-4279
Kinase Inhibitors
>>
VEGFR
Altiratinib (DCC-2701)
AV-951 (Tivozanib)
Cediranib (AZD2171)
Foretinib
MGCD516 (Sitravatinib)
Motesanib (Free base)
Motesanib diphosphate
Pazopanib
Regorafenib
Sunitinib
Vandetanib
Vatalanib
XL184 (Cabozantinib) (free base)
Kinase Inhibitors
>>
WEE1
MK-1775 (Adavosertib) (AZD1775)
Cell Cycle Modulators
>>
Wee1
MK-1775 (Adavosertib) (AZD1775)
Phosphatase Inhibitors/Modulators
>>
Wip1 Phosphatase Inhibitor
GSK2830371
Wnt Signaling Pathway Modulators
C-82
E7386
E-7386
Foscenvivint (PRI-724)
ICG-001
Other Enzyme Inhibitors/Modulators
>>
WRN Helicase Inhibitor
YAP/TAZ Signaling Inhibitor
GNE-7883
IAG933
IK-930
NVP-IAG933
VT-107
Immuno-oncology Modulators
>>
Zinc Finger Protein Degrader
CFT-7455
NVP-DKY709
Special Offers