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BI 6727 (Volasertib)
BI 6727 (Volasertib)
BI6727 (Volasertib)is a highly potent, selective and ATP-competitive inhibitor of polo-like kinases 1 , 2 and 3 (PLK1, 2 and 3), with IC50s at 0.87, 5 and 56 nM, respectively.
Catalog NO:
CT-BI6727
Synonym:
Volasertib
CAS NO:
755038-65-4
Mol. Formula:
C
34
H
50
N
8
O
3
∙0.5H
2
O
MW:
627.8
** in vivo Quality Material. The Optically Pure Source. Hemihydrate, validated by a spot-on Elemental Analysis. Buyers Beware: Partially Racemized BI6727 (with as much as10-30% non-Active Isomer) in marketplace (ref. 3).
Pricing and Ordering
Technical Data
QC & Certificates
References
NO
Size
Price
In Stock
Quantity
1
5 MG
$100.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
2
10 MG
$150.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
3
50 MG
$420.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
4
100 MG
$680.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
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Add To Cart
Solubility :
In DMSO, alcohols, water with 2 eq. of acid
Storage :
Store at 0°C (short term), -20°C (long term), desiccated
Purity :
>99% by Achiral and Chiral HPLCs
Original QC Data :
Achiral and Chiral HPLCs,
1
HNMR and Quantitative Elemental Analysis Report
Please Pick Batch NO:
2
BI-6727, Lot 02, Certificate of Analysis.pdf
BI-6727, Lot 02, Appearance (color).pdf
1. Rudolph, D., et al, BI 6727, a Polo-like kinase inhibitor with improved pharmacokinetic profile and broad antitumor activity, Clin Cancer Res., May 1, 2009; 15 (9), 3094-3102
2. K. Strebhardt, Nature Reviews Drug Discovery, 9, 643-660 (August 2010)
3. with the presence of wrong (Non-Active) isomer (S-Enantiomer) as much as 10-30% from those who fail to report Chiral HPLC Analysis. Only Chiral HPLC separates Active and Non-Active Isomers.
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