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Home > Kinase Inhibitors > RAF (Rapidly Accelerated Fibrosarcoma) > PLX4720

PLX4720

A selective inhibitor of B-RAF protein kinase carrying V600E mutation with a Ki at 13 nM.

Catalog NO:	CT-P4720
Synonym:
CAS NO:	918505-84-7
Mol. Formula:	C₁₇H₁₄ClF₂N₃O₃S
MW:	413.8

** >99.5% (by HPLC at 214 and 254 nm) + A perfect Quantitative Elemental Analysis. Grams in stock from Indianapolis. Ship within 1 day.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	10 mg	$110.00	YES
2	50 mg	$360.00	YES
3	100 mg	$560.00	YES
4	200 mg	$950.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99% (HPLC at 214 and 254 nm)

Original QC Data : LC/MS, ¹HNMR

Please Pick Batch NO:

PLX4720, Lot PL-04, Certificate of Analysis.pdf

1. J. Tsai, et al., Discovery of a selective inhibitor of oncogenic B-Raf kinase with potent antimelanoma activity. Proc Natl Acad Sci USA. 105(8), 3041-6 (2008).

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