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Home > Kinase Inhibitors > BTK (Bruton's Tyrosine Kinase) > Zanubrutinib | BGB-3111

Zanubrutinib | BGB-3111

Zanubrutinib (BGB-3111) is an orally active, potent and selective irreversible Bruton tyrosine kinase (BTk) inhibitor with IC₅₀ = 0.3 nM (ref 1).

Catalog NO:	CT-ZANU
Synonym:	BGB3111
CAS NO:	1691249-45-2
Mol. Formula:	C27H29N5O3
MW:	471.6 (or refer to the Certificate of Analysis, batch-specific)

** in vivo Quality Material. >99% Pure by Achiral and Chiral HPLCs (attached). Anhydrous, verified by a spot-on Elemental Analysis. Bulk stock (Discounted price for 0.5G, 1G, 2G, …). Same Day Shipping

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NO	Size	Price	In Stock	Quantity
1	10 mg	$120.00	YES
2	50 mg	$360.00	YES
3	100 mg	$490.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, NMR, and Elemental Analysis Report

There is no COA file for this product

1. Y. H. Guo, et al., Discovery of Zanubrutinib (BGB-3111), a Novel, Potent, and Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase, J. Med. Chem. 2019, 62, 17, 7923–7940

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