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Home > Kinase Inhibitors > ALK (Anaplastic Lymphoma Kinase) > CEP-28122 Mesylate

CEP-28122 Mesylate

CEP-28122 mesylate is a highly potent, selective and orally active ALK inhibitor (Ezymatic IC50: 1.9 nM (ref 1), 3 nM (ref 2), Cellular IC50: 30 nM (ref 2), Cellular IC50 in 75% murine: 300 nM (ref 2)), displaying a favorable pharmaceutical and pharmacokinetic profile and robust and selective pharmacologic efficacy against ALK-positive human cancer cells and tumor xenograft models in mice.

Catalog NO:	CT-CEPM
Synonym:
CAS NO:	1354545-57-5
Mol. Formula:	C₂₈H₃₅ClN₆O₃ ∙ 1.6CH₄O₃S
MW:	692.8

** in vivo Quality Material. - >99% Pure by Achiral and Chiral HPLCs (Attached). Bulk stock. Same Day Shipping.

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NO	Size	Price	In Stock	Quantity
1	10 mg	$160.00	YES
2	50 mg	$450.00	YES
3	100 mg	$725.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : 100% optical purity (Chiral HPLC), >99% purity (HPLC at 214 and 254 nm)

Original QC Data : HPLC-MS, ¹HNMR, Chiral HPLC, and Quantitative Elemental Analysis

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Current Lot, Certificate of Analysis
C_K, CEP-28122 Mesylate, Lot 01, HPLC-MS.pdf
C_K, CEP-28122 Mesylate, Lot 01, Chiral HPLC.pdf
C_K, CEP-28122 Mesylate, Lot 01, NMR (1-1).pdf

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