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Home > Adenosine Receptor Ligands > Vipadenant

Vipadenant

Vipadenant (BIIB-014) is an orally active, potent and selective adenosine A_2A receptor antagonist with K_i value of 1.3nM, selective over A₁, A_2B and A_A3 receptors (K_is = 68, 63 and 1005 nM, respectively) (ref 1).

Catalog NO:	CT-VIPA
Synonym:	BIIB-014
CAS NO:	442908-10-3
Mol. Formula:	C16H15N7O
MW:	321.3

** >98.5% Pure by HPLC. Anhydrous, verified by a spot-on high-precision Quantitative Microanalysis. Bulk stock! Same day shipping.

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NO	Size	Price	In Stock	Quantity
1	5 mg	$100.00	YES
2	25 mg	$340.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >98.5% by HPLC

Original QC Data : HPLC, NMR, and Quantitative Elemental Analysis

Please Pick Batch NO:

Vipadenant (BIIB-014) Lot 01 Certificate of Analysis.pdf

1. R. J. Gillespie, et al. Antagonists of the human A2A adenosine receptor. 4. Design, synthesis, and preclinical evaluation of 7-aryltriazolo[4,5-d]pyrimidines. J. Med. Chem. 52(1), 33-47 (2009).

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