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GSK046 (iBET-BD2) is a domain-selective and orally active inhibitor of BET with immunomodulatory activity, targeting specifically BDII (Bromodomain II) with IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively (ref 1).
Catalog NO: CT-GSK046
Synonym: iBET-BD2
CAS NO: 2474876-09-8
Mol. Formula: C23H27FN2O4
MW: 414.5
** >98.5% by Achiral and Chiral HPLCs. A single Enantiomer (100% by Chiral HPLC). Monohydrate, validated by a spot-on Quantitative Elemental Analysis. In stock, prompt