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Home > Kinase Inhibitors > CHK (Checkpoint Kinase) > ART-446

ART-446

ART-446 is a potent small molecule CHK2 (Checkpoint kinase 2) inhibitor (IC ₅₀ = 9 nM). It exhibits promising potential in enhancing the therapeutic effects of Olaparib and Irinotecan.

Catalog NO:	CT-ART446
Synonym:	ART446
CAS NO:	2984543-29-3
Mol. Formula:	C20H19F5N8O
MW:	482.4

** in vivo Quality Material. >99% by Achiral and Chiral HPLCs (Attached). Validated Absolute Configuration. Bulk stock (Discounted price for 0.5G, 1G, 2G,…). Same day shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	10 mg	$150.00	YES
2	50 mg	$450.00	YES
3	100 mg	$700.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, MS, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

ART-446 Lot 01 Certificate of Analysis.pdf
ART-446 Lot 01 Visual Appearance .pdf

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