VE-822 (Berzosertib) - Chemietek

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Home > Kinase Inhibitors > ATR (Ataxia Telangiectasia and Rad3 Related) > VE-822 (Berzosertib)

VE-822 (Berzosertib)

VE-822 (Berzosertib, M6620, VX-970) is a potent and selective ATR Kinase inhibitor with a Ki value of 0.2 nM, highly selective over closely-related ATM Kinase (Ki=34 nM, >150 fold selectvity), DNA-PK (Ki >4 uM) and mTOR (Ki >1 uM).

Catalog NO:	CT-VE822
Synonym:	Berzosertib, M6620, VX-976
CAS NO:	1232416-25-9
Mol. Formula:	C₂₄H₂₅N₅O₃S
MW:	463.6

** 99.4% Pure, in vivo Quality material. A yellow crystalline solid, re-crystallized. Anhydrous, validated with a spot-on quantitative elemental analysis. In stock, prompt.

Pricing and OrderingTechnical Data

QC & Certificates

References

NO	Size	Price	In Stock	Quantity
1	10 mg	$110.00	YES
2	50 mg	$295.00	YES
3	100 mg	$475.00	YES
4	200 mg	$775.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99.5% (HPLC at 214 and 254 nm)

Original QC Data : HPLC, ¹HNMR, and Quantitative Elemental Analysis

Please Pick Batch NO:

VE-822, Lot 02, Certificate of Analysis.pdf

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