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NIK (NF-κB-inducing kinase) Inhibitors
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Factor VIIa inhibitor
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TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
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Wee1
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Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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PLK1 (Polo-like Kinase 1) Selective
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RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
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Wee1
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Immunoproteasome Inhibitor
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OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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MTH1 (NUDT1, Human MutT Homologue)
MTH1
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SDAM (Serotonin-Dopamine Activity Modulator)
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
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HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
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p53 Reactivator
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SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
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PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
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Zinc Finger Protein (IKZF1/3) Degrader
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HDAC (histone deacetylase) Inhibitors
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Belinostat
Belinostat
A histone deacetylase (HDAC) inhibitor currently in clinical trial.
Catalog NO:
CT-BELI
Synonym:
PDX101
CAS NO:
414864-00-9
Mol. Formula:
C
1
5
H
1
4
N
2
O
4
S
MW:
318.4
** A clean product with elemental analysis. Ship within 1 day.
Pricing and Ordering
Technical Data
QC & Certificates
References
NO
Size
Price
In Stock
Quantity
1
10 mg
$80.00
YES
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10
2
50 mg
$240.00
YES
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9
10
3
100 mg
$400.00
YES
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8
9
10
4
200 mg
$650.00
YES
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9
10
Bulk Inquiry:
(Contact Us)
Toll-free: 1-877-343-6578 (US and Canada only)
Phone: 317-598-0828;
Email: sales@chemietek.com;
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Solubility :
In DMSO
Storage :
Store at 0°C (short term), -20°C (long term), desiccated
Purity :
99% (HPLC)
Original QC Data :
LC/MS,
1
HNMR
Please Pick Batch NO:
1
Belinostat, Lot 01, Certificate of Analysis.pdf
1. Mackay HJ, Hirte H, Colgan T, Covens A, Macalpine K, Grenci P, Wang L, Mason J, Pham PA, Tsao MS, Pan J, Zwiebel J, Oza AM. Phase II trial of the histone deacetylase inhibitor belinostat in women with platinum resistant epithelial ovarian cancer and micropapillary (LMP) ovarian tumours. Eur J Cancer. 2010 Mar 19. [Epub ahead of print].
2. Paoluzzi L, Scotto L, Marchi E, Zain J, Seshan VE, O'Connor OA. Romidepsin and belinostat synergize the antineoplastic effect of bortezomib in mantle cell lymphoma. Clin Cancer Res. 2010 Jan 15; 16(2):554-65.
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