CT-7001 (Samuraciclib) ( ICEC0942) - Chemietek

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Home > Kinase Inhibitors > CDK (Cyclin-dependent Kinase) > CT-7001 (Samuraciclib) ( ICEC0942)

CT-7001 (Samuraciclib) ( ICEC0942)

CT-7001 (ICEC0942) (Samuraciclib) is a potent, selective and orally bioavailable CDK7 (Cyclin-Dependent Kinase 7) inhibitor, and is currently under evaluation for potential therapies for breast, small-cell lung and haematological cancers.

Catalog NO:	CT-CT7001
Synonym:	ICEC0942, Samuraciclib
CAS NO:	1805789-54-1 (HCl) 1805833-75-3 (Free Base)
Mol. Formula:	C23H30N6O ·2HCl
MW:	479.4 (or, refer to Certificate of Analysis, batch-specific)

** in vivo Quality Material. >99% Pure by achiral and chiral HPLCs (attached), a stereomerically pure single isomer (Validated by Chiral HPLC). HCl salt, validated by an Elemental Analysis. Bulk (Grams), Prompt.

Pricing and OrderingTechnical Data

QC & Certificates

References

NO	Size	Price	In Stock	Quantity
1	5 mg	$125.00	YES
2	10 mg	$175.00	YES
3	50 mg	$495.00	YES
4	100 mg	$895.00	YES

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Solubility : In water, 100mM.

Storage : Refer to Certificate of Analysis

Purity : >99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, MS, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

CT-7001, Lot 01, Certificate of Analysis.pdf
CT-7001, Lot 01, Visual Appearance .pdf

E. K. Ainscow, et al, CT7001: An orally bioavailable CDK7 inhibitor is a potential therapy for breast, small-cell lung and haematological cancers [abstract]. In: Proceedings of the American Association for Cancer Research Annual Meeting 2018; 2018 Apr 14-18; Chicago, IL. Philadelphia (PA): AACR; Cancer Res 2018;78(13 Suppl):Abstract nr 4834.

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