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Home > Kinase Inhibitors > CDK (Cyclin-dependent Kinase) > Enitociclib | (S)-BAY-1251152

Enitociclib | (S)-BAY-1251152

Enitociclib ((S)-Enantiomer, the clinical isomer) ((S)-BAY-1251152, VIP152) is the next-generation, potent and highly selective CDK9/P-TEFb inhibitor.

Catalog NO:	CT-ENITO
Synonym:	(S)-(+)-BAY-1251152, VIP152
CAS NO:	1610408-97-3
Mol. Formula:	C19H18F2N4O2S
MW:	404.4 (or refer to the Certificate of Analysis, batch-specific)

** in vivo Quality Material. 99.5% pure by Achiral and Chiral HPLCs (Attached). Anhydrous, validated by a spot-on Elemental Analysis. Bulk stock (discounted price for 0.5G, 1G, 2G, …). Same day shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	5 mg	$150.00	YES
2	10 mg	$200.00	YES
3	50 mg	$600.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : 99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, MS, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

Enitociclib Lot 01 Certificate of Analysis .pdf
Enitociclib Lot 01 Visual Appearance.pdf
C_K, Enitociclib Lot 01 Achiral HPLC.pdf
C_K, Enitociclib Lot 01 Chiral HPLC.pdf

1. U. Lücking, et al., Changing for the Better: Discovery of the Highly Potent and Selective CDK9 Inhibitor VIP152 Suitable for Once Weekly Intravenous Dosing for the Treatment of Cancer, J Med Chem, 2021, 64 (15): 11651-11674.

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