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BMS-986158 (BMS986158)
BMS-986158 is an orally bioavailable, potent and domain-selective BET protein inhibitor, binding to the acetyl-lysine binding site of BET bromodomain of BRD4 (Bromodomain-containing 4) with an IC50 < 5nM (FRET) (ref. 1). Display excellent pharmacokinetic properties and efficacy in vitro and in vivo antitumor activity. It is currently in clinical evaluation for advanced solid tumor treatment.
Catalog NO: CT-BMS986
Synonym: BMS986158
CAS NO: 1800340-40-2
Mol. Formula: C30H33N5O2
MW: 495.6
** in vivo Grade Material. >99.5% Pure by achiral and chiral HPLCs. A white crystalline powder with a spot-on quantitative microanalysis (element counts). Clean and impeccable (QC Docs attached). Bulk stock! Prompt.