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EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR

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Lysine specific demethylase 1 (LSD1) Inhibitor

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PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators

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Endothelin receptor antagonist (type A specific)

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HMG-CoA reductase inhibitor

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Mutant-IDH1 Inhibitor

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IMPDH Inhibitor

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Liver X receptor (LXR) Agonist/Modulator

RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist

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Toll-like Receptor Agonist

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Anti-angiogenesis

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Arginase Inhibitor

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Prostanoid ligand

RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE

TGFβ Kinase Inhibitor

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Adenosine 2A Receptor Antagonist

Arginase Inhibitor

CD73 (ecto-5'-nucleotidase) Inhibitor

CBP/β-catenin Modulators

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IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor

Zinc Finger Protein Degrader

Immunoproteasome Inhibitor

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mTOR inhibitors

PD-1/PD-L1 CHECKPOINT INHIBITORS

PI3Kγ (GAMMA) Specific Inhibitors

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RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist

SHP2 Phosphatase Inhibitor

STING (Stimulator of Interferon Genes) Agonist

SUMOylation Inhibitor

TGFβ Kinase Inhibitor

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Topoisomerase I

Topoisomerase II

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Kinesin (CENP-E) Inhibitor

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KRAS-PDEδ Interaction Inhibitor

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Tri-complex KRASG12C (ON) Inhibitor

Tri-complex KRAS inhibitors

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Arginase Inhibitor

Glutaminase Inhibitor

IDH (Isocitrate Dehydrogenase) Inhibitors

IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor

MAT2A Inhibitor

Monocarboxylate Transporter 1 (MCT 1) Inhibitor

Monocarboxylate Transporter 4 (MCT 4)

OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator

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Monocarboxylate Transporter 1 (MCT 1) Inhibitor

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Neuroactive/BBB Penetrant

Orexin Receptor Antagonists

SDAM (Serotonin-Dopamine Activity Modulator)

TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor

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CBP/β-catenin Modulators

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Notch Signaling Inhibitors

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CRM1 (exportin 1) Inhibitor(s)

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HCV Protease Inhibitor

HIV-1 integrase Inhibitor

Oxidoreductase Inhibitor

P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor

Thymidylate synthase inhibitor

WRN Helicase Inhibitor

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p53–MDM2 Interaction Inhibitor

p53 Reactivator

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PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors

SHP2 Phosphatase Inhibitor

Wip1 Phosphatase Inhibitor

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PARP (Poly (ADP-ribose) polymerase)

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Stem cell research

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NADD8-Activating Enzyme Inhibtor

Proteasome Inhibitor

SUMOylation Inhibitor

Ubiquitin-Activating Enzyme Inhibitor

USP1 (Ubiquitin Specific Protease 1)

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Home > Hippo Pathway Signaling Inhibitor > IK-930

IK-930

IK-930 is an orally active potent Hippo pathway inhibitor that selectively binds TEAD1 and broadly suppresses oncogenic TEAD signaling.

Catalog NO:	CT-IK930
Synonym:
CAS NO:	2563892-44-2
Mol. Formula:	C19H19F3N4O2S
MW:	424.1

** in vivo Quality Material. 99.5% Pure by HPLC (attached). Anhydrate, validated by a spot-on Elemental Analysis. Bulk stock (Discounted price for 0.2, 0.5, 1G, …). Same Day Shipping.

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NO	Size	Price	In Stock	Quantity
1	10 mg	$100.00	YES
2	50 mg	$300.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : .>99% by HPLC

Original QC Data : HPLC, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

IK-930 Lot 01 Certificate of Analysis.pdf
C_K, IK-930, Lot 01, HPLC.pdf
C_K, IK-930, Lot 01, NMR.pdf

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