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Home > Kinase Inhibitors > PI3K - p110 Alpha (α) Specific > PIK-75

PIK-75

A specific inhibitor of PI3K p110α isoform with IC50 values (nM) of 7.8 (p110α), 343 (p110β), and 907 (p110δ).

Catalog NO:	CT-PIK75
Synonym:
CAS NO:	372196-67-3
Mol. Formula:	C₁₆H₁₄BrN₅O₄S • HCl
MW:	488.75

** Please ask for quote for other quantities.

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NO	Size	Price	In Stock	Quantity
1	10 mg	$70.00	YES
2	50 mg	$180.00	YES
3	100 mg	$300.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99% (HPLC at 214 and 254 nm)

Original QC Data : LC/MS, ¹HNMR

Please Pick Batch NO:

PIK-75, Current Lot, Certificate of Analysis

1. Z. A. Knight, et al., A Pharmacological Map of the PI3-K Family Defines a Role for p110α in Insulin Signaling, Cell 125, 733–747 (2006).

2. C. Chaussade, et al. Evidence for functional redundancy of class IA PI3K isoforms in insulin signaling, Biochem J. 404(3), 449–458 (2007).

3. S. Kim, et al. Insulin-like growth factor-1 regulates platelet activation through PI3-Kα isoform, Blood, 110(13), 4206-4213 (2007).

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