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Kinase Inhibitors
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Syk (Spleen Tyrosine Kinase)
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GS-9973 (Entospletinib)
GS-9973 (Entospletinib)
Spleen tyrosine kinase (Syk), a non-receptor cytoplasmic, BCR-associated enzyme, is expressed in hematopoietic tissues and is often overexpressed in hematopoeitic malignancies. GS-9973 (Entospletinib) is a highly selective and orally efficacious inhibitor of spleen tyrosine kinase (Syk) with an IC50 of 7.7 nM. It inhibits the activity of Syk, which inhibits B-cell receptor (BCR) signaling and leads to an inhibition of tumor cell activation, migration, adhesion and proliferation. It is currently in clinical evaluation for autoimmune and oncology indications.
Catalog NO:
CT-GS9973
Synonym:
Entospletinib
CAS NO:
1229208-44-9
Mol. Formula:
C
23
H
21
N
7
O
MW:
411.5
** A recrystallized crystalline powder/flakes (see attached picture), clean (>99% by HPLC), + impeccable 1H-NMR, coming with a perfect Quantitative Elemental Analysis. Bulk in stock. Ship within 1 day.
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Technical Data
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References
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10 mg
$80.00
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2
50 mg
$160.00
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100 mg
$260.00
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Solubility :
Soluble in DMSO
Storage :
Store at 0°C (short term), -20°C (long term), desiccated
Purity :
>99% Purity (HPLC, detected at 214 and 254 nm)
Original QC Data :
HPLC-MS,
1
HNMR, and Quantitative Elemental Analysis
Please Pick Batch NO:
1
GS-9973, Curent Lot, Certificate of Analysis
GS-9973, Current Lot, NMR
GS-9973, Current Lot, HPLC-MS
GS-9773, Lot 01, Appearance (color).pdf
1. K. S. Currie, et al., Discovery of GS-9973, a Selective and Orally Efficacious Inhibitor of Spleen Tyrosine Kinase, J. Med. Chem., April 6, 2014
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