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Home > Hydrolase Inhibitors/Modulators > Cathepsin K Inhibitor > Odanacatib

Odanacatib

A potent and selective inhibitor of cysteine protease cathepsin K (IC50 0.2 nM), discriminating against cathepsin B (1034 nM), L (2995 nM), and S (60 nM). The product Odanacatib has been in clinical evaluation as the first-in-class drug treating postmenopausal women with osteoporosis.

Catalog NO:	CT-CG001
Synonym:	MK-0822
CAS NO:	603139-19-1
Mol. Formula:	C₂₅H₂₇F₄N₃O₃S ∙ 0.1H₂O
MW:	527.4

** in vivo Quality Material, >99% by Achiral and Chiral HPLCs, with quantitative elemental analysis. White powder. Bulk Stock! Same day shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	10 mg	$130.00	YES
2	50 mg	$250.00	YES
3	100 mg	$425.00	YES
4	200 mg	$750.00	YES

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Solubility : Soluble in DMSO, Alcohols, Common Organic Solvents

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99.8% chem and optical purity (HPLC and chiral HPLC at 214 and 254 nm)

Original QC Data : HPLC-MS, ¹HNMR, Chiral HPLC, and Quantitative Elemental Analysis

Please Pick Batch NO:

Odanacatib, Current Lot, Certificate of Analysis
C_T, Odanacatib, Lot ON001A, LC-MS.pdf
C_T, Odanacatib, Lot ON001A, Chiral HPLC.pdf
C_T, Odanacatib, Lot ON001A, NMR.pdf

1. J. Y. Gauthier, et al, Bioorganic & Medicinal Chemistry Letters (2008), 18 (3), 923 – 928.

* Perfect HPLC, Chiral HPLC, NMR + Quantitative Elemental Analysis + appearance (snow-white powder) , no impurities (not a bit) visible by any analytical methods - a true testament to the superior quality.

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