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Home > Kinase Inhibitors > PI3K - p110 Delta (δ) Specific > IC-87114

IC-87114

IC-87114 is a potent and ATP-competitive PI3K p110δ isoform-selective inhibitor (IC50 = 60 nM). It Inhibits p110α, p110β and p110γ only at much higher concentrations. It does not inhibit other PIK-related kinases such as ATM, ATR, DNA-PK, and mTOR even at concentrations up to 100 µM.

Catalog NO:	CT-IC871
Synonym:	IC87114
CAS NO:	371242-69-2
Mol. Formula:	C₂₂H₁₉N₇O ∙ 0.2H₂O
MW:	401

** A snow-white powder, clean (99.5% by HPLC) + impeccable NMR, with an excellent Quantitative Elemental Analysis, made for animal studies. Bulk in stock. Ship within 1 day.

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NO	Size	Price	In Stock	Quantity
1	10 mg	$85.00	YES
2	50 mg	$200.00	YES
3	100 mg	$350.00	YES
4	200 mg	$600.00	YES
5	500 mg	$1,100.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99.5% (HPLC at 214 and 254 nm)

Original QC Data : HPLC-MS, ¹HNMR, and Quantitative Elemental Analysis

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IC-87114, Current Lot, Certificate of Analysis

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