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Home > KRAS Pathway Inhibitors > G12D Mutant Inhibitors > RMC-9805 | Zoldonrasib

RMC-9805 | Zoldonrasib

Zoldonrasib (RMC-9805) is a first-in-class, mutant-selective, covalent and orally bioavailable tricomplex KRAS ^G12D (ON) inhibitor (refs. 1, 2).

Catalog NO:	CT-RMC9805
Synonym:	Zoldonrasib, RMC9805
CAS NO:	2922732-54-3
Mol. Formula:	C63H88F3N11O7
MW:	1168.4

** in vivo Quality Material. >99% Purity by Achiral and Chiral HPLCs (attached). Hydrate, verified by a spot-on Elemental Analysis. Bulk stock (Discounted price for 0.2, 0.5G, …). Same Day Shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	5 mg	$300.00	YES
2	10 mg	$450.00	YES
3	50 mg	$1,350.00	YES
4	100 mg	$2,250.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

RMC-9805 (Zoldonrasib) Lot 02 Certificate of Analysis.pdf
RMC-9805 Lot 02 Visual Appearance.pdf
C_K, RMC-9805, Lot 02, Achiral HPLC.pdf
C_K, RMC-9805, Lot 02, Chiral HPLC.pdf

1. Knox, J et al.RMC-9805, a first-in-class, mutant-selective, covalent and orally bioavailable KRASG12D(ON) inhibitor, promotes cancer-associated neoantigen recognition and synergizes with immunotherapy in preclinical models. Cancer Res 1 April 2023; 83 (7_Supplement): 3475

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