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Home > Kinase Inhibitors > Glucokinase > MK-0941 Mesylate

MK-0941 Mesylate

MK-0941 Mesylate is an oral allosteric glucokinase activator with EC50 values of 0.24 and 0.065 µM at low (2.5 mM) and high (10 mM) concentrations of glucose, respectively (ref 1). It increases insulin secretion from isolated rat islets of Langerhans and glucose uptake by hepatocytes in vitro. MK-0941 reduces blood glucose levels in high-fat diet-fed db/db mice and in high-fat diet-fed mice with diabetes induced by streptozotocin.

Catalog NO:	CT-MK0941
Synonym:
CAS NO:	1137916-97-2
Mol. Formula:	C21H24N4O6S • CH3SO3H
MW:	556.6

** in vivo Quality Material. >99% by Achiral and Chiral HPLCs (attached). Bulk Stock (Discounted price for 0.2, 0.5, 1, 2G, …,). Same day shipping.

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NO	Size	Price	In Stock	Quantity
1	10 mg	$120.00	YES
2	50 mg	$360.00	YES
3	100 mg	$600.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : 99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, NMR, and Quantitative Elemental Analysis Report

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MK-0941 Mesylate Lot 01 Certificate of Analysis.pdf
C_K, MK-0941 Mesylate, Lot 01, Achiral HPLC.pdf
C_K, MK-0941 Mesylate, Lot 01, Chiral HPLC.pdf

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