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IMPDH Inhibitor

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Arginase Inhibitor

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Prostanoid ligand

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Arginase Inhibitor

Glutaminase Inhibitor

IDH (Isocitrate Dehydrogenase) Inhibitors

IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor

MAT2A Inhibitor

Monocarboxylate Transporter 1 (MCT 1) Inhibitor

Monocarboxylate Transporter 4 (MCT 4)

OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator

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Monocarboxylate Transporter 1 (MCT 1) Inhibitor

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Neuroactive/BBB Penetrant

Orexin Receptor Antagonists

SDAM (Serotonin-Dopamine Activity Modulator)

TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor

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CRM1 (exportin 1) Inhibitor(s)

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HCV Protease Inhibitor

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Oxidoreductase Inhibitor

P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor

Thymidylate synthase inhibitor

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p53–MDM2 Interaction Inhibitor

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PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors

SHP2 Phosphatase Inhibitor

Wip1 Phosphatase Inhibitor

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PARP (Poly (ADP-ribose) polymerase)

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Stem cell research

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NADD8-Activating Enzyme Inhibtor

Proteasome Inhibitor

SUMOylation Inhibitor

Ubiquitin-Activating Enzyme Inhibitor

USP1 (Ubiquitin Specific Protease 1)

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Home > Kinase Inhibitors > PDGFR > Sunitinib

Sunitinib

Sunitinib (SU-11248, Sutent) is an orally available small molecule inhibitor targeting at least eight receptor protein-tyrosine kinases including vascular endothelial growth factor receptors 1–3 (VEGFR1–VEGFR3), platelet-derived growth factor receptors (PDGFRα and PDGFRβ), stem cell factor receptor (Kit), Flt-3, and colony-stimulating factor-1 receptor (CSF-1R).

Catalog NO:	CT-ST001
Synonym:	SU-11248, Sutent
CAS NO:	557795-19-4
Mol. Formula:	C22H27FN4O2
MW:	398.5

** in vivo Quality Material, >99%, anhydrous, validated by a spot-on Quantitative microanalysis. Bulk stock, same day shipping.

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NO	Size	Price	In Stock	Quantity
1	100 mg	$80.00	YES
2	500 mg	$220.00	YES

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Solubility : refer to Certificate of Analysis

Storage : refer to Certificate of Analysis

Purity : >99% by HPLC

Original QC Data : HPLC, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

Sunitinib, Lot ST-1C, Certificate of Analysis.pdf

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