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Home > Kinase Inhibitors > TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase) > Entrectinib

Entrectinib

Entrectinib (RXDX-101, NMS-E628) is an orally available and potent small molecule inhibitor of TrkA, TrkB and TrkC, as well as ROS1 and ALK, with IC50s at lower nanomolar concentrations.

Catalog NO:	CT-ENTR
Synonym:	RXDX-101, NMS-E628
CAS NO:	1108743-60-7
Mol. Formula:	C31H34F2N6O2
MW:	506.6

** in vivo quality material, >99.5% pure, anhydrous, validated by a spot-on quantitative microanalysis. Bulk stock, same day shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	50 mg	$130.00	YES
2	200 mg	$390.00	YES
3	500 mg	$790.00	YES

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Solubility : refer to Certificate of Analysis

Storage : refer to Certificate of Analysis

Purity : >99% by HPLC

Original QC Data : HPLC, NMR, and Elemental Analysis Report

Please Pick Batch NO:

Entrectinib, Lot 01, Certificate of Analysis.pdf

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