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Brexpiprazole (OPC-34712)
Brexpiprazole is a serotonin-dopamine activity modulator (SDAM). Brexpiprazole acts as a partial agonist of the 5-HT1A. D2, and D3 receptors. Partial agonists have both blocking properties and stimulating properties at the receptor they bind to. The ratio of blocking activity to stimulating activity determines a portion of its clinical effects. Brexpiprazole has more blocking and less stimulating activity than its predecessor, aripiprazole, which may decrease its risk for agitation and restlessness. It is also an antagonist of the 5-HT2A, 5-HT2B, 5-HT7, α1A-, α1B-, α1D-, and α2C-adrenergic, and H1 receptors [Ref 1]. It has negligible affinity for the mACh receptors [Ref 1].
Catalog NO: CT-BREX
Synonym: OPC-34712
CAS NO: 913611-97-9
Mol. Formula: C25H27N3O2S
MW: 433.6
** A snow-white crystalline powder, >99.5% pure, coming with a perfect quantitative elemental analysis. Bulk stock. Ship within 1 day.