TAK-788 (Mobocertinib) - Chemietek

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Home > Kinase Inhibitors > EGFR Mutants > TAK-788 (Mobocertinib)

TAK-788 (Mobocertinib)

TAK-788 (Mobocertinib, AP32788) is a potent and selective covalent inhibitor targeting EGFR and human EGFR 2 (HER2) exon 20 insertion mutations, with minimal inhibitory activity against Wt-EGFR. It has been granted Breakthrough Therapy Designation by FDA for the treatment of lung cancer with HER2 mutations or EGFR mutations including exon 20 insertion mutations.

Catalog NO:	CT-TAK788
Synonym:	Mobocertinib, AP32788
CAS NO:	1847461-43-1
Mol. Formula:	C32H39N7O4
MW:	585.7

** 99.5% Pure. in vivo Quality Material. Clean and impeccable (Data Attached). Anhydrous, salt-free, validated by a spot-on Elemental Analysis. Bulk Stock (Get quote for 10G, 20G). Prompt..

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NO	Size	Price	In Stock	Quantity
1	10 mg	$75.00	YES
2	50 mg	$160.00	YES
3	200 mg	$450.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% by HPLC

Original QC Data : HPLC-MS, 1H-NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

TAK-788, Lot 01, Certificate of Analysis.pdf
TAK-788, Lot 01, Visual Appearance .pdf
C_K, TAK-788, Lot 01, HPLC-MS (1).pdf
C_K, TAK-788, Lot 01, NMR in DMSO (1-2).pdf

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