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Akt/(PKB (Protein Kinase B)
ALK (Anaplastic Lymphoma Kinase)
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ASK1 (Apoptosis Signal-regulating Kinase 1)
ATM (Ataxia Telangiectasia Mutated Kinase)
ATR (Ataxia Telangiectasia and Rad3 Related)
Aurora Kinase
Aurora A Kinase Selective
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Aurora C Kinase Selective
AXL (AXL Receptor Tyrosine Kinase)
Bcr-Abl/c-kit/PDGFR/Src
BTK (Bruton's Tyrosine Kinase)
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CDK (Cyclin-dependent Kinase)
CDK2 Selective
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EGFR Mutants
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EphB4 (Ephrin Type-B Receptor 4) Kinase
ErbB
Erk (Extracellular signal regulated kinase)
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FLT3 (Fms-like Tyrosine Kinase 3)
IGF-1R
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LRRK2
MEK/MAPK
Mps1 (Monopolar Spindle 1)
mTOR
NIK (NF-κB-inducing kinase) Inhibitors
P21-Activated Kinases
P70S6K (Ribosomal Protein S6 Kinase)
PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
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PKMYT1
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PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
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ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
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TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
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WEE1
Factor VIIa inhibitor
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Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
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PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
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Prostanoid ligand
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Tri-complex KRAS inhibitors
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IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
MTH1
Neuroactive/BBB Penetrant
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PARP (Poly (ADP-ribose) polymerase)
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AXL (AXL Receptor Tyrosine Kinase)
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BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
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c-Met
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ErbB
Erk (Extracellular signal regulated kinase)
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PDK1
PI3K - p110 Alpha (α) Specific
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PI3K/mTOR
PIM
PKC (Protein Kinase C)
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
PLK4 (Polo-like Kinase 4) Selective
PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
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WEE1
Activated Factor VII (Factor VIIa)
Factor VIIa inhibitor
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PRC2 (the catalytic subunit of polycomb repressive complex 2) >
PKMYT1 Kinase Inhibitor
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TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Tubulin
Wee1
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CoreDAC Inhibitors
DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
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EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
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Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
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PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
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PLA2 Inhibitors
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IDH (Isocitrate Dehydrogenase) Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
IMPDH Inhibitor
Immune Activation Agents/Modulators
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Arginase Inhibitor
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Prostanoid ligand
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TGFβ Kinase Inhibitor
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Immuno-oncology Modulators
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IKZF1/3 (Zinc Finger Protein 1/3)
Immunoproteasome Inhibitor
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mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
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PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
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Tri-complex KRAS inhibitors
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Metabolic Pathway Modulators
Arginase Inhibitor
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IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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MTH1 (NUDT1, Human MutT Homologue)
MTH1
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SDAM (Serotonin-Dopamine Activity Modulator)
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
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CBP/β-catenin Modulators
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Notch Signaling Inhibitors
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HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Interaction Inhibitor/Modulator
p53–MDM2 Interaction Inhibitor
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PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
PLA2 (Phospholipase A2) Inhibitor
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PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
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Varespladib Methyl (LY333013)
Varespladib Methyl (LY333013)
Varespladib methyl is a secretory phospholipase A2 (sPLA2) inhibitor. It is an orally bioavailable prodrug of the varespladib, currently in clinical evaluation.
Catalog NO:
CT-VAREM
Synonym:
A-002, LY333013, S-3013
CAS NO:
172733-08-3
Mol. Formula:
C
2
2
H
2
2
N
2
O
5
MW:
394.4
** 99.9% pure. in vivo Quality Material. Textbook quality (see all attached QC docs). Bulk stock. Same day shipping.
Pricing and Ordering
Technical Data
QC & Certificates
References
NO
Size
Price
In Stock
Quantity
1
10 mg
$120.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
2
50 mg
$320.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
3
100 mg
$490.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
4
200 mg
$850.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
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(Contact Us)
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Solubility :
In DMSO (>100MG)
Storage :
Store at 0°C (short term), -20°C (long term), desiccated
Purity :
99.9% (by HPLC at 214 and 254 nm)
Original QC Data :
HPLC,
1
H-NMR, and quantitative elemental analysis report
Please Pick Batch NO:
2
Varespladib Methyl, Lot 02, Certificate of Analysis.pdf
C_K, Varespladib Methyl, Lot 02, HPLC.pdf
C_K, Varespladib Methyl, Lot 02, NMR.pdf
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Unit Price
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