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Home > Adenosine Receptor Ligands > SCH442416

SCH442416

SCH442416 is a potent and selective adenosine A_2A receptor antagonist. Binds to human and rat A_2A receptors with high affinity (K_i values are 0.05 and 0.5 nM respectively). Displays > 23000-fold selectivity for hA_2A over hA₁ in vitro with minimal affinity for hA_2B and hA₃ receptors (IC₅₀ > 10 μM).

Catalog NO:	CT-SCH442
Synonym:	SCH-442416
CAS NO:	316173-57-6
Mol. Formula:	C20H19N7O2
MW:	389.4

** in vivo Quality Material. >99% Pure by HPLC, Anhydrous, verified by a spot-on high-precision Quantitative Microanalysis. Bulk stock! Same day shipping.

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NO	Size	Price	In Stock	Quantity
1	5 mg	$130.00	YES
2	25 mg	$480.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : 99% by HPLC

Original QC Data : HPLC, NMR, and Quantitative Elemental Analysis

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SCH442416 Lot 01 Certificate of Analysis.pdf

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