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Home > Kinase Inhibitors > FGFR (Fibroblast Growth Factor Receptor) > Erdafitinib (JNJ-42756493)

Erdafitinib (JNJ-42756493)

Erdafitinib (JNJ-42756493) is a first-in-class, orally available, potent and selective pan FGFR family inhibitor, with biochemical IC50 values of 1.2, 2.5, 3, and 5.7 nM for FGFR1-4, respectively. (ref. 1)

Catalog NO:	CT-ERDA
Synonym:	JNJ-42756493
CAS NO:	1346242-81-6
Mol. Formula:	C25H30N6O2
MW:	446.6

** in vivo Quality Material. >99.5% by HPLC. Hemihydrate, Validated by a Quantitative Elemental Analysis. Bulk Stock. Prompt.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	10 mg	$70.00	YES
2	50 mg	$150.00	YES
3	100 mg	$250.00	YES
4	200 mg	$400.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% (HPLC)

Original QC Data : HPLC, NMR and Quantitative Elemental Analysis Report

Please Pick Batch NO:

Erdafitinib, Lot 01, Certificate of Analysis.pdf
Erdafitinib, Lot 01, Visual Appearance.pdf

1. Perera T. P. S, et al, Discovery and pharmacological characterization of JNJ-42756493 (erdafitinib), a functionally selective small molecule FGFR family inhibitor. Mol Cancer Ther. 2017, Vol 16, No 6, P1010-1020

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