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Home > Other Enzyme Inhibitors/Modulators > HCV Protease Inhibitor > VX-950

VX-950

A potent, selective and orally bioavailable inhibitor of hepatitis C virus NS3.4A serine protease, a first hepatitis C drug currently in development that has demonstrated activity in patients who have failed prior therapy.

Catalog NO:	CT-VX950
Synonym:	Telaprevir
CAS NO:	402957-28-2
Mol. Formula:	C₃₆H₅₃N₇O₆
MW:	679.85

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	2 mg	$200.00	YES
2	5 mg	$400.00	YES
3	10 mg	$600.00	YES
4	50 mg	$1,800.00	YES

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Solubility : In DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >98% purity (HPLC)

Original QC Data : LC/MS, ¹HNMR

Please Pick Batch NO:

VX-950, Lot 01, COA
VX-950, Lot 01, NMR
VX-950, Lot 01, LC-MS

1. McHutchison JG, et al., "Telaprevir for previously treated chronic HCV infection". N. Engl. J. Med. (2010) 362 (14): 1292–303

2. Irena Melnikova, "Hepatitis C therapies". Nature Reviews Drug Discovery (2008) 7: 799–800

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