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Home > New Products (II) > RMC-6236

RMC-6236

RMC-6236 is a First-in-Class, non-covalent, oral, potent, and RAS-Selective Tri-Complex RAS^MULTI(ON) Inhibitor with activity across a diverse spectrum of RAS mutants, including KRASG12V and KRASG12D (Ref 1).

Catalog NO:	CT-RMC6236
Synonym:	RMC6236
CAS NO:	2765081-21-6
Mol. Formula:	C44H58N8O5S
MW:	811.0

** in vivo Quality Material. >99% Purity by Achiral and Chiral HPLCs (attached), with a Quantitative Elemental Analysis. Bulk stock (Discounted price for 0.2, 0.5, 1G, …). Same day shipping.

Pricing and OrderingTechnical Data

QC & Certificates

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NO	Size	Price	In Stock	Quantity
1	5 mg	$400.00	YES
2	10 mg	$550.00	YES
3	50mg	$1,700.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

RMC-6236 (RMC6236) Lot 01 Certificate of Analysis.pdf
RMC-6236 Lot 01 Visual Appearance .pdf
C_K, RMC-6236, Lot 01, LC-MS.pdf
C_K, RMC-6236, Lot 01, Chiral HPLC.pdf

1. Elena S. Koltun, et al, Direct targeting of KRASG12X mutant cancers with RMC-6236, a first-in-class, RAS-selective, orally bioavailable, tri-complex RASMULTI(ON) inhibitor [abstract]. In: Proceedings of the American Association for Cancer Research Annual Meeting 2022; 2022 Apr 8-13. Philadelphia (PA): AACR; Cancer Res 2022;82(12_Suppl): Abstract nr 3597.

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