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Home > New Products (II) > FX-909

FX-909

FX-909 is a first-in-class, orally available and highly potent covalent inverse agonist of the peroxisome proliferator-activated receptor gamma (PPARG) lineage transcription factor with cellular IC₅₀ = 1 nM, highly selective over PPARA/PPARD (related transcription factors) (over 2000-fold selectivity).

Catalog NO:	CT-FX909
Synonym:	FX909
CAS NO:	2935964-98-8
Mol. Formula:	C17H10F2N2O3S
MW:	360.3

** in vivo Quality material. 99.9% Pure by HPLC (Attached). Anhydrous, validated by a spot-on Elemental Analysis. Bulk stock (Discounted price for Larger Sizes: 0.2, 0.5, 1, 2G,…,). Same Day Shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	10 mg	$200.00	YES
2	50 mg	$600.00	YES
3	100 mg	$1,000.00	YES
4	200 mg	$1,600.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% by HPLC

Original QC Data : HPLC, MS, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

FX-909, Lot 01, Certificate of Analysis.pdf
FX-909, Lot 01, Visual Appearance.pdf
C_K, FX-909, Lot 01, HPLC.pdf
C_K, FX-909, Lot 01, NMR.pdf

1. R. Sim, et al, Discovery of FX-909, a first-in-class inverse agonist of the peroxisome proliferator-activated receptor gamma (PPARG) lineage transcription factor, to potentially treat patients with the luminal subtype of advanced urothelial cancer (UC) [abstract]. In: Proceedings of the American Association for Cancer Research Annual Meeting 2023; Part 1 (Regular and Invited Abstracts); 2023 Apr 14-19; Orlando, FL. Philadelphia (PA): AACR; Cancer Res 2023;83(7_Suppl):Abstract nr ND08

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