BI-907828 (Brigimadlin) - Chemietek

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Home > Cell Cycle Modulators > p53-MDM2 Interaction Inhibitor > BI-907828 (Brigimadlin)

BI-907828 (Brigimadlin)

Brigimadlin (BI-907828) is an orally bioavailable, highly potent, and selective small molecule inhibitor of the MDM2 and p53 interaction.

Catalog NO:	CT-BRIG
Synonym:	Brigimadlin, BI907828
CAS NO:	2095116-40-6
Mol. Formula:	C31H25Cl2FN4O3
MW:	591.5 (Or refer to the Certificate of Analysis, batch-specific)

** in vivo Quality Material. >99% Pure by Achiral and Chiral HPLCs (attached). Validated Activity (IC₅₀ = 2-3 nM). Hemihydrate, verified by a spot-on Microanalysis. Bulk stock (Discounted price for 0.2, 0.5, 1G, …). Same Day Shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	5 mg	$200.00	YES
2	10 mg	$260.00	YES
3	50 mg	$800.00	YES

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Solubility : Refer to Certificate of Analysis

Storage : Refer to Certificate of Analysis

Purity : >99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

BI-907828, Lot 01, Certificate of Analysis.pdf
BI-907828, Lot 01, Visual Appearance.pdf
C_K, BI-907828, Lot 01, Achiral HPLC.pdf
C_K, BI-907828, Lot 01, Chiral HPLC.pdf

1. Gollner Andreas, et al. Preparation of spiroindolepyrrolidinone derivatives for use as MDM2-p53 inhibitors: World Intellectual Property Organization, WO2017060431. 2017-04-13.

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