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NIK (NF-κB-inducing kinase) Inhibitors
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PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
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PKMYT1
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Factor VIIa inhibitor
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Arginase Inhibitor
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Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
MTH1
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
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PARP (Poly (ADP-ribose) polymerase)
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USP1 (Ubiquitin Specific Protease 1)
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PKC (Protein Kinase C)
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PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
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PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
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Factor VIIa inhibitor
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TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
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Wee1
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DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
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Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
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IDH (Isocitrate Dehydrogenase) Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
IMPDH Inhibitor
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OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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MTH1
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HCV Protease Inhibitor
HIV-1 integrase Inhibitor
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Thymidylate synthase inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
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Wip1 Phosphatase Inhibitor
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Hippo Pathway Signaling Inhibitor
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VT-107
VT-107
VT-107 is a potent and selective TEAD Auto-palmitoylation inhibitor that Inhibits Proliferation and Tumor Growth of NF2-deficient Mesothelioma. VT-107 prevented palmitoylation of the TEAD1 protein, and decreased the levels of palmitoylated TEAD3 and TEAD4.
Catalog NO:
CT-VT107
Synonym:
VT107
CAS NO:
2417718-63-7
Mol. Formula:
C
25
H
20
F
3
N
3
O
MW:
435.5
** in vivo Quality Material. >99% Pure by Achiral and Chiral HPLCs (attached). Hydrate, validated by a spot-on Elemental Analysis. Bulk stock (Discounted price for 0.2, 0.5, 1, 2G, …). Same Day Shipping.
Pricing and Ordering
Technical Data
QC & Certificates
References
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Size
Price
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Quantity
1
5 mg
$100.00
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10 mg
$150.00
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3
50 mg
$450.00
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9
10
4
100 mg
$700.00
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10
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Solubility :
Refer to Certificate of Analysis
Storage :
Refer to Certificate of Analysis
Purity :
>99% by Achiral and Chiral HPLCs
Original QC Data :
Achiral and Chiral HPLCs, MS, NMR, and Quantitative Elemental Analysis Report
Please Pick Batch NO:
1
VT-107, Lot 01, Certificate of Analysis.pdf
VT-107, Lot 01, Visual Appearance.pdf
C_K, VT-107, Lot 01, Achiral HPLC.pdf
C_K, VT-107, Lot 01, Chiral HPLC.pdf
C_K, VT-107, Lot 01, NMR.pdf
1. Tang TT, et al. Small Molecule Inhibitors of TEAD Auto-palmitoylation Selectively Inhibit Proliferation and Tumor Growth of NF2-deficient Mesothelioma. Mol Cancer Ther. 2021; 20(6):986-998.
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