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Home > Kinase Inhibitors > MEK/MAPK > PD-0325901

PD-0325901

PD 0325901(Mirdametinib) is an orally available, potent and highly selective small molecule inhibitor of both MEK1 and MEK2 (MAPK/ERK Kinase) with a Ki value at low nM.

Catalog NO:	CT-PD03
Synonym:	Mirdametinib, PD0325901
CAS NO:	391210-10-9
Mol. Formula:	C₁₆H₁₄F₃IN₂O₄
MW:	482.2

** in vivo Quality material. >99.5% by achiral and Chiral HPLCs (attached). A white powder. Anhydrous, validated by a spot-on quantitative elemental analysis. Bulk stock. Same day shipping.

Pricing and OrderingTechnical Data

QC & Certificates

References

NO	Size	Price	In Stock	Quantity
1	10 mg	$80.00	YES
2	50 mg	$160.00	YES
3	100 mg	$260.00	YES
4	200 mg	$450.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99% Achiral and Chiral HPLCs.

Original QC Data : Achiral, Chiral HPLCs, MS, ¹HNMR, Quantitative Elemental Analysis Report

Please Pick Batch NO:

PD-0325901, Lot 04, Certificate of Analysis.pdf
PD-0325901, Lot 04, Visual Appearance.pdf
C_K, PD0325901, Lot 04, HPLC-MS.pdf
C_K, PD0325901, Lot 04, Chiral HPLC.pdf
C_K, PD0325901, Lot 04, NMR.pdf

1. Barrett, SD et al. “The discovery of the benzhydroxamine MEK inhibitors CI-1040 and PD 0325901” Bioorg. Med. Chem. Lett. 2008, 18, 6501-6504.

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