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Home > Phosphatase Inhibitors/Modulators > SHP2 Phosphatase Inhibitor > JAB-3068

JAB-3068

JAB-3068 is a potent, selective and orally bioavailable allosteric inhibitor of SHP2 (protein tyrosine phosphatase) (PTP) non-receptor type 11 (SHP2; Src homology region 2 domain phosphatase; PTPN11), with potential antineoplastic activity. It is efficacious as an oral monotherapy as well as an immune-oncology modulator.

Catalog NO:	CT-JAB3068
Synonym:	JAB3068
CAS NO:	2169223-48-5
Mol. Formula:	C22H26F2N6O2S
MW:	476.5

** in vivo Quality Material. >99.5% Pure by achiral and chiral HPLCs, an Enantiomerically pure single isomer (100% by Chiral HPLC). Free base (Salt-free), anhydrous, validated by a spot-on microanalysis, made for in vivo studies. Bulk stock, prompt.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	5 mg	$170.00	YES
2	10 mg	$250.00	YES
3	50 mg	$850.00	YES

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Solubility : refer to Certificate of Analysis

Storage : refer to Certificate of Analysis

Purity : >99% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, MS, NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

JAB-3068, Lot 01, Certificate of Analysis.pdf
JAB-3068, Lot 01, Visual Appearance .pdf

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