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ALK (Anaplastic Lymphoma Kinase)
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ASK1 (Apoptosis Signal-regulating Kinase 1)
ATM (Ataxia Telangiectasia Mutated Kinase)
ATR (Ataxia Telangiectasia and Rad3 Related)
Aurora Kinase
Aurora A Kinase Selective
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AXL (AXL Receptor Tyrosine Kinase)
Bcr-Abl/c-kit/PDGFR/Src
BTK (Bruton's Tyrosine Kinase)
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
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ErbB
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IGF-1R
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LRRK2
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Mps1 (Monopolar Spindle 1)
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NIK (NF-κB-inducing kinase) Inhibitors
P21-Activated Kinases
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PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
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PKMYT1
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PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
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ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
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Factor VIIa inhibitor
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Menin-MLL interaction inhibitors
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Arginase Inhibitor
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IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
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Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
MTH1
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
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PARP (Poly (ADP-ribose) polymerase)
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USP1 (Ubiquitin Specific Protease 1)
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PKC (Protein Kinase C)
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
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PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
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TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
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Wee1
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DNMT1 (DNA Methyltransferase 1) inhibitor
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Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
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IDH (Isocitrate Dehydrogenase) Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
IMPDH Inhibitor
Immune Activation Agents/Modulators
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Arginase Inhibitor
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Immunoproteasome Inhibitor
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mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
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IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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MTH1
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TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
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Gamma (γ) Secretase (GS) Inhibitors
Notch Signaling Inhibitors
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HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
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p53 Reactivator
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Wip1 Phosphatase Inhibitor
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PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
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BCL-XL Selective Inhibitors
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DT-2216
DT-2216
DT-2216 is a selective B-cell lymphoma-extra large (Bcl-XL) targeted protein degrader with potential pro-apoptotic, immunomodulating and antineoplastic activities (ref 1).
Catalog NO:
CT-DT2216
Synonym:
CAS NO:
2365172-42-3
Mol. Formula:
C77H96ClF3N10O10S4
MW:
1542.4
** 99% by HPLC. Anhydrous, validated by a spot-on Quantitative Elemental Analysis. In stock, same day shipping.
Pricing and Ordering
Technical Data
QC & Certificates
References
NO
Size
Price
In Stock
Quantity
1
5 mg
$180.00
YES
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9
10
2
25 mg
$620.00
YES
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1
2
3
4
5
6
7
8
9
10
3
50 mg
$980.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
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Solubility :
Refer to Certificate of Analysis
Storage :
Refer to Certificate of Analysis
Purity :
>99% by HPLC
Original QC Data :
HPLC, NMR, and Elemental Analysis Report
Please Pick Batch NO:
1
DT-2216, Lot 01, Certificate of Analysis.pdf
1. Y He, et al. DT2216 - a Bcl-XL-specific degrader is highly active against Bcl-xL-dependent T cell lymphomas. J Hematol Oncol 13, 95 (2020). https://doi.org/10.1186/s13045-020-00928-9
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