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Home > G-Protein-coupled Receptor Ligands > Adenosine Receptor Ligands > CVT-6883

CVT-6883

A potent and highly selective antagonist of A2b adenosine receptor (A2bAR) with a Ki of 8.3 nM, differentiating from other adenosine receptors, such as A1 (~10,000 nM), A2a (>10,000 nM) and A3 (>>10,000 nM).

Catalog NO:	CT-CV001
Synonym:	GS 6201
CAS NO:	752222-83-6
Mol. Formula:	C₂₁H₂₁F₃N₆O₂
MW:	446.4

** Please ask for quote for other quantities.

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NO	Size	Price	In Stock	Quantity
1	10 mg	$150.00	YES
2	50 mg	$490.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >98.5% (HPLC)

Original QC Data : MS (EI), ¹HNMR, HPLC

Please Pick Batch NO:

CVT-6883, Current Lot, COA
CVT-6883, Current Lot, NMR
CVT-6883, Current Lot, HPLC

1. Chun-Xiao Sun, et al, The Journal of Clinical Investigation (August 2006) 116 (8), 2173-2182; 2. Jacobson KA, et al," Nature reviews. Drug discovery (2006) 5 (3), 247-64.

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