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EMD1214063 (Tepotinib)
EMD1214063 (Tepotinib) is an orally bioavailable, potent and selective inhibitor of c-Met, inhibiting the enzyme with an IC50 value of 3 nM, highly selective (≥ 1000-fold) over a panel of 242 other kinases; inhibits c-Met phosphorylation and downstream signaling targets in various cancer cell lines with IC50s of 6-9 nM; demonstrates in vivo antitumor efficacy in mouse xenograft models (ref 1).
Catalog NO: CT-EMD063
Synonym: EMD-1214063, MSC2156119
CAS NO: 1100598-32-0
Mol. Formula: C29H28N6O2
MW: 492.6
** White powder with quantitative elemental analysis. In stock, prompt.