XL184 (Cabozantinib) (free base) - Chemietek

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Home > Kinase Inhibitors > c-Met > XL184 (Cabozantinib) (free base)

XL184 (Cabozantinib) (free base)

XL184 (Cabozantinib) is an orally active, multitargeted inhibitor of tumor growth, metastasis and angiogenesis, simultaneously targeting c-MET, RET and VEGFR2 with IC50s at low nM.

Catalog NO:	CT-XL184
Synonym:	Cabozantinib, BMS907351, BMS-907351
CAS NO:	849217-68-1
Mol. Formula:	C₂₈H₂₄FN₃O₅
MW:	501.5

** A snow-white recrystallized powder (picture attached), clean (>99.5% pure), with a perfect quantitative elemental analysis, for in vivo studies. Bulk Stock! Same day shipping.

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NO	Size	Price	In Stock	Quantity
1	50 MG	$100.00	YES
2	200 MG	$230.00	YES

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Solubility : In DMSO

Storage : 0 °C (short term), -20 °C (long term), Desiccated

Purity : >99.5% (HPLC at 214 and 254 nm)

Original QC Data : ¹HNMR, HPLC/MS, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

XL-184 (Cabozantinib), Lot 03, Certificate of Analysis.pdf
XL184 (Cabozantinib), Lot 03, Visual Appearance (color).pdf

1. Kurzrock, R., et al., J Clin Oncol, 2011 Jul 1; 29(9): 2662-6.

2. Durante, C., et al., Expert Opin Investig Drugs, 2011 May; 20 (3): 403-413

3.You WK, et al. Cancer Res, 2011, 71(14), 4758-4768

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