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Home > Other Enzyme Inhibitors/Modulators > P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor > RX-5902 (Supinoxin)

RX-5902 (Supinoxin)

RX-5902 (Supinoxin) is an orally administered small molecule inhibitor of a unique cancer protein – phosphorylated-p68 RNA Helicase (P-p68), a protein selectively overexpressed in cancer cells and absent in normal tissue. P-p68 is believed to increase the activity of multiple cancer related genes including, cyclin D1, c-jun and c-myc, and plays a prominent role in tumor progression and metastasis. Over-expression of P-p68 has been observed in many solid tumors, including, melanoma, colon, ovarian and lung tumors. RX-5902, as a single agent, inhibits tumor growth and enhances survival in a variety of in vivo animal xenograft tumor models (e.g., renal, ovarian, pancreatic, melanoma).

Catalog NO:	CT-RX5902
Synonym:	Supinoxin
CAS NO:	888478-45-3
Mol. Formula:	C22H24FN5O4
MW:	441.5

** in vivo grade material. Snow-white crystalline powder, 99.9% purity by HPLC + a clean and impeccable 1H-NMR + a spot-on high-precision quantitative elemental analysis. Ship within 1 day from Indianapolis.

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NO	Size	Price	In Stock	Quantity
1	5 mg	$110.00	YES
2	10 mg	$160.00	YES
3	50 mg	$450.00	YES
4	100 mg	$750.00	YES

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Solubility : Refer to Certificate

Storage : Refer to Certificate

Purity : 99.9% by HPLC (at 214 and 254 nm)

Original QC Data : HPLC-MS, 1H-NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

RX-5902,, Lot 01, Appearance (color).pdf
RX-5902, Lot 01, Certificate of Analysis, 1.0.pdf

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