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Home > Kinase Inhibitors > RAF (Rapidly Accelerated Fibrosarcoma) > PLX4032

PLX4032

A selective inhibitor of B-RAF protein kinase carrying V600E mutation with an IC₅₀ of 44 nM.

Catalog NO:	CT-P4032
Synonym:	Vemurafenib, RG7204, RO5185426
CAS NO:	1029872-54-5
Mol. Formula:	C₂₃H₁₈ClF₂N₃O₃S
MW:	489.9

** in vivo Quality Material. >99% Purity, with a spot-on quantitative elemental analysis. Bulk stock. Prompt.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	10 mg	$60.00	YES
2	50 mg	$140.00	YES
3	100 mg	$220.00	YES
4	200 mg	$390.00	YES
5	500 mg	$750.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : 99.5% (HPLC at 214 and 254 nm)

Original QC Data : HPLC-MS, ¹HNMR, and Quantitative Elemental Analysis

Please Pick Batch NO:

PLX4032, Lot 016 (curent Lot),Certificate of Analysis.pdf

1. Bollag, G., et al., Clinical efficacy of a RAF inhibitor needs broad target blockade in BRAF-mutant melanoma, Nature, 467, 596-9 (2010).

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