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IDO1 (INDOLEAMINE 2,3-DIOXYGENASE 1) Inhibitors
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
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OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Interaction Inhibitor/Modulator
PCNA (Proliferating Cell Nuclear Antigen)
PDE4 ( Phosphodiesterase Type 4) Inhibitor/Modulators
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PLA2 (Phospholipase A2) Inhibitor
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PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
Reagents for Biological Assays
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SMAC Mimics and Inhibitors of IAP
Stem Cell Research Products
STING (Stimulator of Interferon Genes) Agonist
SUMO Pathway Modulator
TEAD Inhibitor
Toll-like Receptor Agonist
Ubiquitin / Proteasome System
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YAP/TAZ Signaling Inhibitor
Zinc Finger Protein (IKZF1/3) Degrader
Akt/(PKB (Protein Kinase B)
ALK (Anaplastic Lymphoma Kinase)
AMPK (AMP-Activated Protein Kinase)
ASK1 (Apoptosis Signal-regulating Kinase 1)
ATM (Ataxia Telangiectasia Mutated Kinase)
ATR (Ataxia Telangiectasia and Rad3 Related)
Aurora Kinase
Aurora A Kinase Selective
Aurora B Kinase Selective
Aurora C Kinase Selective
AXL (AXL Receptor Tyrosine Kinase)
Bcr-Abl/c-kit/PDGFR/Src
BTK (Bruton's Tyrosine Kinase)
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CDK (Cyclin-dependent Kinase)
CDK2 Selective
CDK4 Selective
CDK7 Selective
CDK9 Selective
CDK12/CDK13
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
CLK2 (CDC2-like Kinase 2)
c-Met
DDK (Dbf4-dependent kinase)
DNA-PK (DNA-Dependent Protein Kinase)
EGFR Mutants
EGFR/HER2
EphB4 (Ephrin Type-B Receptor 4) Kinase
ErbB
Erk (Extracellular signal regulated kinase)
FAK (Focal Adhesion Kinase)
FGFR (Fibroblast Growth Factor Receptor)
FGFR4 Specific
FLT3 (Fms-like Tyrosine Kinase 3)
IGF-1R
JAK (Janus Kinase)
JAK1 Selective
JAK1/JAK2 Selective
JAK2 Selective
JAK3 Selective
LRRK2
MEK/MAPK
Mps1 (Monopolar Spindle 1)
mTOR
NIK (NF-κB-inducing kinase) Inhibitors
P21-Activated Kinases
P70S6K (Ribosomal Protein S6 Kinase)
PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
PI3K - p110 Beta (β) Specific
PI3K - p110 Delta (δ) Specific
PI3K - p110 Gamma (γ) Specific
PI3K - Pan
PI3K/mTOR
PIM
PKC (Protein Kinase C)
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
PLK4 (Polo-like Kinase 4) Selective
PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
VEGFR
WEE1
Factor VIIa inhibitor
Bcl-2 Family Protein Inhibitors
BCL-2 Selective Inhibitors
BCL-XL Protein Degrader
BCL-XL Selective Inhibitors
MCL-1 Selective Inhibitors
CD73 (ecto-5'-nucleotidase) Inhibitor
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CBP/β-catenin Modulators
Cell Cycle/DNA Damage
CDK Inhibitors/Modulators
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
DNA Replication Modulators/Breakers
Endoplasmic Reticulum Stress Modulator (ERSM)
G-Quadruplex Ligand
IMPDH Inhibitor
Kinesin (CENP-E) Inhibitor
KRAS-G12C Inhibitors
KRASG12C (ON) (Tri-complex) Inhibitor
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KRAS-PDEδ Interaction Inhibitor
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Menin-MLL interaction inhibitors
Mps1 (Monopolar Spindle 1)
Notch Signaling Inhibitors
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
p53-MDM2 Interaction Inhibitor
PCNA (Proliferating Cell Nuclear Antigen)
PRC2 (the catalytic subunit of polycomb repressive complex 2) >
PKMYT1 Kinase Inhibitor
SMAC Mimics and Inhibitors of IAP
Survivin
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Tubulin
Wee1
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Mutant Isocitrate Dehydrogenase-1 (IDH1) Inhibitor
Mutant Isocitrate Dehydrogenase-2 (IDH2) Inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
Chemotherapy Agents
ATPases (BRG1/BRM)
BET Family Protein Degraders
BET Family Protein Inhibitors
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BET/BRD9 Degrader
BET Bromodomain II (BDII) Selective Inhibitors
BET/Domain & Sub-set Selective Inhibitors
CBP/P300 Bromodomain Inhibitor
CoreDAC Inhibitors
DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
EP300/CBP HAT (Histone Acetyltransferases) Inhibitor
EZH1/2 Dual Inhibitors
EZH2 Methyltransferase Inhibitors
EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
HDAC (histone deacetylase) Inhibitors
HDAC1-Specific Inhibitors
HDAC3-Specific Inhibitors
HDAC6-Specific Inhibitors
Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
PRC2 (the catalytic subunit of polycomb repressive complex 2)
PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
PRMTs (Type I) Inhibitors/Modulators
Adenosine Receptor Ligands
Angiotensin II receptor (AT1)
Endothelin receptor antagonist (type A specific)
Heat Shock Proteins HSP90 Inhibitors
Hedgehog Signaling Pathway Inhibitors
HMG-CoA reductase inhibitor
Androgen receptor
Glucocorticoid Receptor
RXRs (retinoid X receptors)
Autotaxin Inhibitor
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Cathepsin K Inhibitor
Neprilysin (MME) Inhibitor
PDE4 ( phosphodiesterase type 4)
PLA2 Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH Inhibitor
Liver X receptor (LXR) Agonist/Modulator
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
STING (STIMULATOR OF INTERFERON GENES) AGONIST
Toll-like Receptor Agonist
Anti-angiogenesis
Anti-fibrosis
Anti-inflammatory
Arginase Inhibitor
Autotaxin Inhibitors
PLA2 Inhibitors
Prostanoid ligand
RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE
TGFβ Kinase Inhibitor
Adenosine 2A Receptor Antagonist
Arginase Inhibitor
CD73 (ecto-5'-nucleotidase) Inhibitor
CBP/β-catenin Modulators
CoreDAC Inhibitors
IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
IKZF1/3 (Zinc Finger Protein 1/3)
Immunoproteasome Inhibitor
Liver X receptor (LXR) Agonist/Modulator
mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
PI3Kγ (GAMMA) Specific Inhibitors
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SHP2 Phosphatase Inhibitor
STING (Stimulator of Interferon Genes) Agonist
SUMOylation Inhibitor
TGFβ Kinase Inhibitor
Toll-like Receptor Agonist
Topoisomerase I
Topoisomerase II
Kinesin (CENP-E) Inhibitor
G12C Mutant Inhibitors
G12D Mutant Inhibitors
KRAS-PDEδ Interaction Inhibitor
Pan-KRAS Inhibitors
SOS1 Inhibitors
Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
MTH1
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
SDAM (Serotonin-Dopamine Activity Modulator)
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
CBP/β-catenin Modulators
Gamma (γ) Secretase (GS) Inhibitors
Notch Signaling Inhibitors
CRM1 (exportin 1) Inhibitor(s)
HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
p53–MDM2 Interaction Inhibitor
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
PARP (Poly (ADP-ribose) polymerase)
Stem cell research
NADD8-Activating Enzyme Inhibtor
Proteasome Inhibitor
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Ubiquitin-Activating Enzyme Inhibitor
USP1 (Ubiquitin Specific Protease 1)
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Akt/(PKB (Protein Kinase B)
ALK (Anaplastic Lymphoma Kinase)
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ATM (Ataxia Telangiectasia Mutated Kinase)
ATR (Ataxia Telangiectasia and Rad3 Related)
Aurora Kinase
Aurora A Kinase Selective
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Aurora C Kinase Selective
AXL (AXL Receptor Tyrosine Kinase)
Bcr-Abl/c-kit/PDGFR/Src
BTK (Bruton's Tyrosine Kinase)
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CDC7 (Cell Division Cycle 7-related Protein Kinase)
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CDK2 Selective
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CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
CLK2 (CDC2-like Kinase 2)
c-Met
DDK (Dbf4-dependent kinase)
DNA-PK (DNA-Dependent Protein Kinase)
EGFR Mutants
EGFR/HER2
EphB4 (Ephrin Type-B Receptor 4) Kinase
ErbB
Erk (Extracellular signal regulated kinase)
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FGFR4 Specific
FLT3 (Fms-like Tyrosine Kinase 3)
IGF-1R
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mTOR
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P70S6K (Ribosomal Protein S6 Kinase)
PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
PI3K - p110 Beta (β) Specific
PI3K - p110 Delta (δ) Specific
PI3K - p110 Gamma (γ) Specific
PI3K - Pan
PI3K/mTOR
PIM
PKC (Protein Kinase C)
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
PLK4 (Polo-like Kinase 4) Selective
PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
VEGFR
WEE1
Activated Factor VII (Factor VIIa)
Factor VIIa inhibitor
Arginase Inhibitor
Adenosine Receptor Ligands
Autotaxin Inhibitor
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Bcl-2 Family Protein Inhibitors
BCL-2 Selective Inhibitors
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MCL-1 Selective Inhibitors
BCL-6 Protein Inhibitors
CD73 Immune Pathway Inhibitor/Modulator
CD73 (ecto-5'-nucleotidase) Inhibitor
Cell Cycle Modulators
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CBP/β-catenin Modulators
Cell Cycle/DNA Damage
CDK Inhibitors/Modulators
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
DNA Replication Modulators/Breakers
Endoplasmic Reticulum Stress Modulator (ERSM)
G-Quadruplex Ligand
IMPDH Inhibitor
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KRAS-PDEδ Interaction Inhibitor
KRAS-SOS1 Inhibitors
Menin-MLL interaction inhibitors
Mps1 (Monopolar Spindle 1)
Notch Signaling Inhibitors
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
p53-MDM2 Interaction Inhibitor
PCNA (Proliferating Cell Nuclear Antigen)
PRC2 (the catalytic subunit of polycomb repressive complex 2) >
PKMYT1 Kinase Inhibitor
SMAC Mimics and Inhibitors of IAP
Survivin
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Tubulin
Wee1
Cell Metabolism Modulators
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Mutant Isocitrate Dehydrogenase-1 (IDH1) Inhibitor
Mutant Isocitrate Dehydrogenase-2 (IDH2) Inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
Chemotherapy
Chemotherapy Agents
CoREST-selective Deacetylase (CoreDAC) inhibitors
Degraders (Protein Degraders)
DNA Methyltransferase Inhibtors
DNA Repair Targeted Therapy
DNA/RNA Synthesis Inhibitor/Blocker
Endoplasmic Reticulum Stress Modulator (ERSM)
Epigenetics Resch Products
ATPases (BRG1/BRM)
BET Family Protein Degraders
BET Family Protein Inhibitors
BET/Bromodomain (BDI and BDII) Selective Inhibitors
BET/BRD4 Degrader
BET/BRD9 Degrader
BET Bromodomain II (BDII) Selective Inhibitors
BET/Domain & Sub-set Selective Inhibitors
CBP/P300 Bromodomain Inhibitor
CoreDAC Inhibitors
DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
EP300/CBP HAT (Histone Acetyltransferases) Inhibitor
EZH1/2 Dual Inhibitors
EZH2 Methyltransferase Inhibitors
EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
HDAC (histone deacetylase) Inhibitors
HDAC1-Specific Inhibitors
HDAC3-Specific Inhibitors
HDAC6-Specific Inhibitors
Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
PRC2 (the catalytic subunit of polycomb repressive complex 2)
PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
PRMTs (Type I) Inhibitors/Modulators
Gamma (γ) Secretase (GS) Inhibitors
Glucocorticoid Receptor Antagonist/Modulator
Glutaminase Inhibitor
G-Protein-coupled Receptor Ligands
Adenosine Receptor Ligands
Angiotensin II receptor (AT1)
Endothelin receptor antagonist (type A specific)
Heat Shock Protein Research Products
Heat Shock Proteins HSP90 Inhibitors
Hedgehog Signaling Pathway Modulators
Hedgehog Signaling Pathway Inhibitors
Hippo Pathway Signaling Inhibitor
HMG-CoA Reductase
HMG-CoA reductase inhibitor
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Androgen receptor
Glucocorticoid Receptor
RXRs (retinoid X receptors)
Hydrolase Inhibitors/Modulators
Autotaxin Inhibitor
Caspase-1 Inhibitor
Cathepsin K Inhibitor
Neprilysin (MME) Inhibitor
PDE4 ( phosphodiesterase type 4)
PLA2 Inhibitors
IDO1 (INDOLEAMINE 2,3-DIOXYGENASE 1) Inhibitors
IDH (Isocitrate Dehydrogenase) Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
IMPDH Inhibitor
Immune Activation Agents/Modulators
Liver X receptor (LXR) Agonist/Modulator
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
STING (STIMULATOR OF INTERFERON GENES) AGONIST
Toll-like Receptor Agonist
Immuno/Inflammatory Mediators
Anti-angiogenesis
Anti-fibrosis
Anti-inflammatory
Arginase Inhibitor
Autotaxin Inhibitors
PLA2 Inhibitors
Prostanoid ligand
RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE
TGFβ Kinase Inhibitor
Immunoproteasome Inhibitor
Immuno-oncology Modulators
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Arginase Inhibitor
CD73 (ecto-5'-nucleotidase) Inhibitor
CBP/β-catenin Modulators
CoreDAC Inhibitors
IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
IKZF1/3 (Zinc Finger Protein 1/3)
Immunoproteasome Inhibitor
Liver X receptor (LXR) Agonist/Modulator
mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
PI3Kγ (GAMMA) Specific Inhibitors
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SHP2 Phosphatase Inhibitor
STING (Stimulator of Interferon Genes) Agonist
SUMOylation Inhibitor
TGFβ Kinase Inhibitor
Toll-like Receptor Agonist
Immunosuppressants/Immunochemotherapy Agents
Isomerase Inhibitor/Modulator
Topoisomerase I
Topoisomerase II
Kinesin Ligand/Modulator
Kinesin (CENP-E) Inhibitor
KRAS Pathway Inhibitors
G12C Mutant Inhibitors
G12D Mutant Inhibitors
KRAS-PDEδ Interaction Inhibitor
Pan-KRAS Inhibitors
SOS1 Inhibitors
Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Liver X receptor (LXR) Agonist/Modulator
Metabolic Pathway Modulators
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4) Inhibitor
MTH1 (NUDT1, Human MutT Homologue)
MTH1
Neuroactive Research Products
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
SDAM (Serotonin-Dopamine Activity Modulator)
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
Notch/Wnt Signaling Pathway
CBP/β-catenin Modulators
Gamma (γ) Secretase (GS) Inhibitors
Notch Signaling Inhibitors
Nuclear Export Protein Inhibitors/Modulators
CRM1 (exportin 1) Inhibitor(s)
Other Enzyme Inhibitors/Modulators
HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Interaction Inhibitor/Modulator
p53–MDM2 Interaction Inhibitor
PCNA (Proliferating Cell Nuclear Antigen)
PDE4 ( Phosphodiesterase Type 4) Inhibitor/Modulators
Phosphatase Inhibitors/Modulators
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
PLA2 (Phospholipase A2) Inhibitor
Polymerase Inhibitor/Modulator
PARP (Poly (ADP-ribose) polymerase)
PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
Reagents for Biological Assays
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SMAC Mimics and Inhibitors of IAP
Stem Cell Research Products
Stem cell research
STING (Stimulator of Interferon Genes) Agonist
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TEAD Inhibitor
Toll-like Receptor Agonist
Ubiquitin / Proteasome System
NADD8-Activating Enzyme Inhibtor
Proteasome Inhibitor
SUMOylation Inhibitor
Ubiquitin-Activating Enzyme Inhibitor
USP1 (Ubiquitin Specific Protease 1)
Wnt Signaling Pathway Modulators
YAP/TAZ Signaling Inhibitor
Zinc Finger Protein (IKZF1/3) Degrader
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Anti-fibrosis
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Pirfenidone
Pirfenidone
Pirfenidone is a well-established antifibrotic and anti-inflammatory agent both in vitro and in vivo. It inhibits TGF-β stimulated collagen production, and reduces the production of fibrogenic mediators such as TGF-β and inflammatory mediators such as TNF-α and IL-1β.
Catalog NO:
CT-PIRF
Synonym:
Esbriet, Pirespa, Etuary
CAS NO:
53179-13-8
Mol. Formula:
C12H11NO
MW:
185.2
** in vivo Quality Material. >99% by HPLC + clean NMR + a spot-on quantitative elemental analysis. Pale yellow crystals. Bulk quantities in stock. Ship within 1 day.
Pricing and Ordering
Technical Data
QC & Certificates
References
NO
Size
Price
In Stock
Quantity
1
50 mg
$75.00
YES
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2
200 mg
$150.00
YES
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9
10
3
500 mg
$225.00
YES
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9
10
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Solubility :
In DMSO
Storage :
refer to COA
Purity :
>99 (HPLC at 214 and 254 nm)
Original QC Data :
HPLC-MS, NMR and Quantitative Elemental Analysis
Please Pick Batch NO:
1
Pirfenidone, Lot 01, Certificate of Analysis.pdf
C_K, Pirfenidone, Lot 01, HPLC-MS.PDF
C_K, Pirfenidone, Lot 01, NMR.pdf
Pirfenidone, Lot 01, Visual Appearance .pdf
1. CJ Schaefer, et al, Antifibrotic activities of pirfenidone in animal models, Eur Respir Rev, June 2011, 20 (120): 85–97
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