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IDO1 (INDOLEAMINE 2,3-DIOXYGENASE 1) Inhibitors
IDH (Isocitrate Dehydrogenase) Inhibitors
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PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Interaction Inhibitor/Modulator
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PLA2 (Phospholipase A2) Inhibitor
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Reagents for Biological Assays
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SMAC Mimics and Inhibitors of IAP
Stem Cell Research Products
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Zinc Finger Protein (IKZF1/3) Degrader
Akt/(PKB (Protein Kinase B)
ALK (Anaplastic Lymphoma Kinase)
AMPK (AMP-Activated Protein Kinase)
ASK1 (Apoptosis Signal-regulating Kinase 1)
ATM (Ataxia Telangiectasia Mutated Kinase)
ATR (Ataxia Telangiectasia and Rad3 Related)
Aurora Kinase
Aurora A Kinase Selective
Aurora B Kinase Selective
Aurora C Kinase Selective
AXL (AXL Receptor Tyrosine Kinase)
Bcr-Abl/c-kit/PDGFR/Src
BTK (Bruton's Tyrosine Kinase)
BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
CDC7 (Cell Division Cycle 7-related Protein Kinase)
CDK (Cyclin-dependent Kinase)
CDK2 Selective
CDK4 Selective
CDK7 Selective
CDK9 Selective
CDK12/CDK13
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
CLK2 (CDC2-like Kinase 2)
c-Met
DDK (Dbf4-dependent kinase)
DNA-PK (DNA-Dependent Protein Kinase)
EGFR Mutants
EGFR/HER2
EphB4 (Ephrin Type-B Receptor 4) Kinase
ErbB
Erk (Extracellular signal regulated kinase)
FAK (Focal Adhesion Kinase)
FGFR (Fibroblast Growth Factor Receptor)
FGFR4 Specific
FLT3 (Fms-like Tyrosine Kinase 3)
IGF-1R
JAK (Janus Kinase)
JAK1 Selective
JAK1/JAK2 Selective
JAK2 Selective
JAK3 Selective
LRRK2
MEK/MAPK
Mps1 (Monopolar Spindle 1)
mTOR
NIK (NF-κB-inducing kinase) Inhibitors
P21-Activated Kinases
P70S6K (Ribosomal Protein S6 Kinase)
PDGFR
PDK1
PI3K - p110 Alpha (α) Specific
PI3K - p110 Beta (β) Specific
PI3K - p110 Delta (δ) Specific
PI3K - p110 Gamma (γ) Specific
PI3K - Pan
PI3K/mTOR
PIM
PKC (Protein Kinase C)
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
PLK4 (Polo-like Kinase 4) Selective
PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
VEGFR
WEE1
Factor VIIa inhibitor
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CD73 (ecto-5'-nucleotidase) Inhibitor
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CBP/β-catenin Modulators
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CDC7 (Cell Division Cycle 7-related Protein Kinase)
CHK (Checkpoint Kinase)
CLK (CDC2-like-Kinase)
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Endoplasmic Reticulum Stress Modulator (ERSM)
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IMPDH Inhibitor
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Menin-MLL interaction inhibitors
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PRC2 (the catalytic subunit of polycomb repressive complex 2) >
PKMYT1 Kinase Inhibitor
SMAC Mimics and Inhibitors of IAP
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TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Tubulin
Wee1
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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BET/Domain & Sub-set Selective Inhibitors
CBP/P300 Bromodomain Inhibitor
CoreDAC Inhibitors
DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
EP300/CBP HAT (Histone Acetyltransferases) Inhibitor
EZH1/2 Dual Inhibitors
EZH2 Methyltransferase Inhibitors
EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
HDAC (histone deacetylase) Inhibitors
HDAC1-Specific Inhibitors
HDAC3-Specific Inhibitors
HDAC6-Specific Inhibitors
Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
PRC2 (the catalytic subunit of polycomb repressive complex 2)
PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
PRMTs (Type I) Inhibitors/Modulators
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STING (STIMULATOR OF INTERFERON GENES) AGONIST
Toll-like Receptor Agonist
Anti-angiogenesis
Anti-fibrosis
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Arginase Inhibitor
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Prostanoid ligand
RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE
TGFβ Kinase Inhibitor
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Arginase Inhibitor
CD73 (ecto-5'-nucleotidase) Inhibitor
CBP/β-catenin Modulators
CoreDAC Inhibitors
IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
IKZF1/3 (Zinc Finger Protein 1/3)
Immunoproteasome Inhibitor
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mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
PI3Kγ (GAMMA) Specific Inhibitors
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SHP2 Phosphatase Inhibitor
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SUMOylation Inhibitor
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Kinesin (CENP-E) Inhibitor
G12C Mutant Inhibitors
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SOS1 Inhibitors
Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
MTH1
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
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Thymidylate synthase inhibitor
p53–MDM2 Interaction Inhibitor
PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
PARP (Poly (ADP-ribose) polymerase)
Stem cell research
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USP1 (Ubiquitin Specific Protease 1)
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BUB1 (Budding Uninhibited by Benzimidazoles 1)(Mitotic checkpoint serine/threonine-protein kinase)
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ErbB
Erk (Extracellular signal regulated kinase)
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PDK1
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PI3K/mTOR
PIM
PKC (Protein Kinase C)
PKMYT1
PLK (Polo-like kinase)
PLK1 (Polo-like Kinase 1) Selective
PLK4 (Polo-like Kinase 4) Selective
PTEF-b/CDK9
RAF (Rapidly Accelerated Fibrosarcoma)
RET (Rearranged During Transfection) Kinase
RIP1 (Receptor Interacting Protein 1) Kinase
ROCK (Rho-Associated Protein Kinase)
ROS1 (Proto-oncogene Tyrosine-protein Kinase ROS)
Syk (Spleen Tyrosine Kinase)
TGFβ (Transforming Growth Factor Beta (TGFβ) Receptor) Kinase
TOPK (T–lymphokine-activated killer cell–originated protein kinase)
TRK (Tropomyosin Receptor Kinase) (Tyrosine Receptor Kinase)
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
VEGFR
WEE1
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Factor VIIa inhibitor
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CBP/β-catenin Modulators
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CLK (CDC2-like-Kinase)
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G-Quadruplex Ligand
IMPDH Inhibitor
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Menin-MLL interaction inhibitors
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Notch Signaling Inhibitors
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator/Inhibitor
p53-MDM2 Interaction Inhibitor
PCNA (Proliferating Cell Nuclear Antigen)
PRC2 (the catalytic subunit of polycomb repressive complex 2) >
PKMYT1 Kinase Inhibitor
SMAC Mimics and Inhibitors of IAP
Survivin
TTK (Human Protein Kinase Monopolar Spindle 1 (hMps1))
Tubulin
Wee1
Cell Metabolism Modulators
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
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Chemotherapy
Chemotherapy Agents
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CBP/P300 Bromodomain Inhibitor
CoreDAC Inhibitors
DNMT1 (DNA Methyltransferase 1) inhibitor
DOT1L Methyltransferase Inhibitor
EP300/CBP HAT (Histone Acetyltransferases) Inhibitor
EZH1/2 Dual Inhibitors
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EZH2 (Mutant) METHYLTRANSFERASE INHIBITOR
HDAC (histone deacetylase) Inhibitors
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Lysine specific demethylase 1 (LSD1) Inhibitor
Menin-MLL interaction inhibitors
PRC2 (the catalytic subunit of polycomb repressive complex 2)
PRMT5 (Protein Arginine Methyltransferase 5) Inhibitors/Modulators
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Endothelin receptor antagonist (type A specific)
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HMG-CoA reductase inhibitor
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IDH (Isocitrate Dehydrogenase) Inhibitors
Mutant-IDH1 Inhibitor
Mutant-IDH2 Inhibitor
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
IMPDH Inhibitor
Immune Activation Agents/Modulators
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STING (STIMULATOR OF INTERFERON GENES) AGONIST
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Arginase Inhibitor
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Prostanoid ligand
RIP1 (RECEPTOR INTERACTING PROTEIN 1) KINASE
TGFβ Kinase Inhibitor
Immunoproteasome Inhibitor
Immuno-oncology Modulators
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CD73 (ecto-5'-nucleotidase) Inhibitor
CBP/β-catenin Modulators
CoreDAC Inhibitors
IDO1 (Indoleamine 2,3-dioxygenase 1) Inhibitor
IKZF1/3 (Zinc Finger Protein 1/3)
Immunoproteasome Inhibitor
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mTOR inhibitors
PD-1/PD-L1 CHECKPOINT INHIBITORS
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PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SHP2 Phosphatase Inhibitor
STING (Stimulator of Interferon Genes) Agonist
SUMOylation Inhibitor
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Tri-complex KRASG12C (ON) Inhibitor
Tri-complex KRAS inhibitors
Liver X receptor (LXR) Agonist/Modulator
Metabolic Pathway Modulators
Arginase Inhibitor
Glutaminase Inhibitor
IDH (Isocitrate Dehydrogenase) Inhibitors
IMPDH (Inosine Monosphosphate Dehydrogenase) Inhibitor
MAT2A Inhibitor
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4)
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
Monocarboxylate Transporter 1 (MCT 1) Inhibitor/Ligand
Monocarboxylate Transporter 1 (MCT 1) Inhibitor
Monocarboxylate Transporter 4 (MCT 4) Inhibitor
MTH1 (NUDT1, Human MutT Homologue)
MTH1
Neuroactive Research Products
Neuroactive/BBB Penetrant
Orexin Receptor Antagonists
SDAM (Serotonin-Dopamine Activity Modulator)
TRK (Tropomyosin Receptor Kinase)(Tyrosine Receptor Kinase) Inhibitor
Notch/Wnt Signaling Pathway
CBP/β-catenin Modulators
Gamma (γ) Secretase (GS) Inhibitors
Notch Signaling Inhibitors
Nuclear Export Protein Inhibitors/Modulators
CRM1 (exportin 1) Inhibitor(s)
Other Enzyme Inhibitors/Modulators
HCV Protease Inhibitor
HIV-1 integrase Inhibitor
Oxidoreductase Inhibitor
P-p68 (Phosphorylated-p68 RNA Helicase) Inhibitor
Thymidylate synthase inhibitor
OXPHOS (Mitochondrial Oxidative Phosphorylation of Complex I) Modulator
PD-1/PD-L1 Checkpoint Inhibitors
p53–MDM2 Interaction Inhibitor/Modulator
p53–MDM2 Interaction Inhibitor
PCNA (Proliferating Cell Nuclear Antigen)
PDE4 ( Phosphodiesterase Type 4) Inhibitor/Modulators
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PTPN2/N1 (Protein Tyrosine Phosphatase Non-Receptor Type 2/1) Inhibitors
SHP2 Phosphatase Inhibitor
Wip1 Phosphatase Inhibitor
PLA2 (Phospholipase A2) Inhibitor
Polymerase Inhibitor/Modulator
PARP (Poly (ADP-ribose) polymerase)
PPARG Agonist (Peroxisome Proliferator-activated Receptor Gamma Agomist)
Reagents for Biological Assays
RORγ (Retinoic Acid-related Orphan Receptor gamma (γ )) Agonist
SMAC Mimics and Inhibitors of IAP
Stem Cell Research Products
Stem cell research
STING (Stimulator of Interferon Genes) Agonist
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Ubiquitin / Proteasome System
NADD8-Activating Enzyme Inhibtor
Proteasome Inhibitor
SUMOylation Inhibitor
Ubiquitin-Activating Enzyme Inhibitor
USP1 (Ubiquitin Specific Protease 1)
Wnt Signaling Pathway Modulators
YAP/TAZ Signaling Inhibitor
Zinc Finger Protein (IKZF1/3) Degrader
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c-Met
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PF-04217903
PF-04217903
A potent, selective (>1000-fold more selective than other 208 kinases), orally bioavailable c-Met kinase inhibitor with Ki at low nM.
Catalog NO:
CT-PF0421
Synonym:
CAS NO:
956905-27-4
Mol. Formula:
C
1
9
H
1
6
N
8
O
MW:
372.38
** in vivo Quality material. 99% Pure by HPLC (Attached). Anhydrous, validated by a spot-on Elemental Analysis. Bulk stock. Same day shipping.
Pricing and Ordering
Technical Data
QC & Certificates
References
NO
Size
Price
In Stock
Quantity
1
10 mg
$100.00
YES
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1
2
3
4
5
6
7
8
9
10
2
50 mg
$300.00
YES
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1
2
3
4
5
6
7
8
9
10
3
100 mg
$490.00
YES
--Select--
1
2
3
4
5
6
7
8
9
10
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Solubility :
Soluble in DMSO, water (pH < 7)
Storage :
Store at 0°C (short term), -20°C (long term), desiccated
Purity :
≥ 99% (HPLC)
Original QC Data :
LC/MS,
1
HNMR
Please Pick Batch NO:
1
PF-04217903^J Lot 01^J Certificate of Analysis.pdf
1. S. L. Timofeevski, et al, Enzymatic Characterization of c-Met Receptor Tyrosine Kinase Oncogenic Mutants and Kinetic Studies with Aminopyridine and Triazolopyrazine Inhibitors, Biochemistry, 2009, 48 (23), 5339–5349.
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