PD-1 Inhibitor 16 (Aurigene Compound 16) - Chemietek

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Home > Immunosuppressants/Immunochemotherapy Agents > PD-1 Inhibitor 16 (Aurigene Compound 16)

PD-1 Inhibitor 16 (Aurigene Compound 16)

PD-1 Inhibitor 16 (Aurigene Compound 16) (extracted from Patent (compound 16, ref 1)) is an orally bioavailable small molecule peptidomimetic inhibitor of the immune checkpoint regulatory proteins PD-I/PD-L1 (programmed cell death -1/programmed cell death ligand-1) interaction, with signaling activity in cancer cells, and is currently being evaluated as a potential negative immune checkpoint regulatory and antineoplastic agent.

Catalog NO:	CT-PD1-16
Synonym:
CAS NO:	2005454-12-4
Mol. Formula:	C14H23N7O6∙H2O
MW:	403.4 (or refer to Certificate of Analysis, batch-specific)

** in vivo grade material, >99.5% purity (HPLC at 214nm), Snow-white powder (picture attached), monohydrate.* In stock. Same day shipping.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	5 mg (Exact Weight)	$190.00	YES
2	10 mg (Exact Weight)	$280.00	YES
3	50 mg (Exact Weight)	$1,050.00	YES

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Solubility : refer to Certificate of Analysis

Storage : refer to Certificate of Analysis

Purity : >99.5% by HPLC (at 214 nm)

Original QC Data : HPLC, 1H-NMR, Quantitative Elemental Analysis Report

Please Pick Batch NO:

PD1 Inhibitor 16, Lot 01, Visual Appearance.pdf
PD1 Inhibitor 16, Lot 01, Certificate of Anal.pdf

1. Patent WO2016142886, 3-SUBSTITUTED-1,2,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS

*Validated by a high-precision quantitative elemental analysis.

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