Sapanisertib (TAK-228) (MLN0128) - Chemietek

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Home > Kinase Inhibitors > mTOR > Sapanisertib (TAK-228) (MLN0128)

Sapanisertib (TAK-228) (MLN0128)

Sapanisertib (TAK-228) (MLN0128) is a potent, selective, orally bioavailable and ATP-competitive mTORC1/C2 inhibitor with an IC50 at low nM, currently in clinical trials.

Catalog NO:	CT-INK128
Synonym:	Sapanisertib, TAK-228, MLN0128, INK128
CAS NO:	1224844-38-5
Mol. Formula:	C₁₅H₁₅N₇O
MW:	309.3

** in vivo grade material. A clean product with >99.5% purity + a spot-on quantitative elemental analysis + validated bioactivity (In-house assay for the product has yielded IC50 at 1 - 1.2 nM for mTORC1/C2). Bulk, prompt.

Pricing and OrderingTechnical Data

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NO	Size	Price	In Stock	Quantity
1	10 mg	$120.00	YES
2	50 mg	$275.00	YES
3	100 mg	$490.00	YES
4	200 mg	$750.00	YES

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Solubility : In DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99.5% (HPLC at 215 and 254 nm)

Original QC Data : HPLC-MS, ¹HNMR, and Quantitative Elemental Analysis

Please Pick Batch NO:

INK128, Current Lot, Certificate of Analysis

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