CORT125134 (Relacorilant) ( CORT-125134) - Chemietek

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Home > Glucocorticoid Receptor Antagonist/Modulator > CORT125134 (Relacorilant) ( CORT-125134)

CORT125134 (Relacorilant) ( CORT-125134)

CORT125134 (Relacorilant) is an orally active next generation high‐affinity antagonist of the glucocorticoid receptor (GR) with high selectivity over other steroid receptors. It is currently being evaluated, in combination with other standard care of agent(s), for treatment of endogenous Cushing's syndrome, and other forms of solid tumors.

Catalog NO:	CT-CORT12
Synonym:	Relacorilant, CORT-125134
CAS NO:	1496510-51-0
Mol. Formula:	C27H22F4N6O3S
MW:	586.6

** in vivo Quality material. 99.7-100% by achiral and chiral HPLCs (All Qc docs attached), coming with a spot-on quantitative microanalysis. Bulk stock!! Prompt shipping.

Pricing and OrderingTechnical Data

QC & Certificates

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NO	Size	Price	In Stock	Quantity
1	5 mg	$200.00	YES
2	10 mg	$300.00	YES
3	50 mg	$960.00	YES

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Solubility : refer to Certificate of Analysis

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : 99.7-100% by Achiral and Chiral HPLCs

Original QC Data : Achiral and Chiral HPLCs, MS, 1H-NMR, and Quantitative Elemental Analysis Report

Please Pick Batch NO:

CORT125134 (Relacorilant), Lot 01, Certificate of Analysis.pdf
CORT125134 (Relacorilant), Lot 01, Visual Appearance.pdf
C_K, CORT-125134, Lot 01, Achiral HPLC.pdf
C_K, CORT-125134, Lot 01, Chiral HPLC.pdf
C_K, CORT-125134, Lot 01, NMR, (1-1).pdf

1. H. Hunt, et al, Preclinical efficacy of the selective GR antagonist, CORT125134, in: Proceedings of the American Association for Cancer Research Annual Meeting 2017; 2017 Apr 1-5; Washington, DC. Philadelphia (PA): AACR; Cancer Res 2017;77(13 Suppl):Abstract nr 3623. doi:10.1158/1538-7445. AM2017-3623

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