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Home > Kinase Inhibitors > ALK (Anaplastic Lymphoma Kinase) > CH5424802

CH5424802

CH5424802 is a potent, selective and orally bioavailable Anaplastic Lymphoma Kinase (ALK) Inhibitor (IC₅₀ = 1.9 nM) capable of blocking the resistant gatekeeper mutant.

Catalog NO:	CT-CH542
Synonym:	Alectinib
CAS NO:	1256580-46-7
Mol. Formula:	C₃₀H₃₄N₄O₂∙0.5HCl∙0.5H₂O
MW:	509.9

** Grams in stock, coming with an excellent quantitative elemental analysis. Ship within 1 day.

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NO	Size	Price	In Stock	Quantity
1	5 mg	$100.00	YES
2	10 mg	$150.00	YES
3	50 mg	$450.00	YES
4	100 mg	$750.00	YES

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Solubility : In DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99% (HPLC at 214 and 254 nm)

Original QC Data : HPLC-MS, ¹HNMR, and Quantitative Elemental Analysis

Please Pick Batch NO:

CH5424802, Current, COA

1. H. Sakamoto, et al., Cancer Cell, Volume 19, Issue 5, p679-690

2. K. Kinoshita, et al., Design and synthesis of a highly selective, orally active and potent anaplastic lymphoma kinase inhibitor. Bioorganic & Medicinal Chemistry, Vol. 20, Issue 3, 1 February 2012, Pages 1271-1280

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