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Home > Polymerase Inhibitor/Modulator > PARP (Poly (ADP-ribose) polymerase) > BSI-201

BSI-201

A selective, irreversible and orally bioavailable inhibitor of poly(ADPribose) polymerase-1 (PARP-1), currently in clinical trial (phase III) for cancer therapy.

Catalog NO:	CT-BSI201
Synonym:	Iniparib
CAS NO:	160003-66-7
Mol. Formula:	C₇H₅IN₂O₃
MW:	292.03

** Please ask for quote for other quantities. Yellow crystalline powder. Grams in stock.

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NO	Size	Price	In Stock	Quantity
1	50 mg	$50.00	YES
2	200 mg	$120.00	YES
3	500 mg	$200.00	YES

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Solubility : Soluble in DMSO, and alcohols

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : > 99% (HPLC)

Original QC Data : HPLC, MS and ¹HNMR

There is no COA file for this product

1. Pal SK, Childs BH, Pegram M. Triple negative breast cancer: unmet medical needs. Breast Cancer Res Treat. 2010 Dec 15. [Epub ahead of print] PubMed PMID: 21161370.

2. Liang H, Tan AR. Iniparib, a PARP1 inhibitor for the potential treatment of cancer, including triple-negative breast cancer. IDrugs. 2010 Sep; 13(9):646-56.

3. He JX, Yang CH, Miao ZH. Poly(ADP-ribose) polymerase inhibitors as promising cancer therapeutics. Acta Pharmacol Sin. 2010 Sep; 31(9):1172-80.

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