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Home > Ubiquitin / Proteasome System > Proteasome Inhibitor > Bortezomib

Bortezomib

A potent and highly selective inhibitor of 20S proteasome with a Ki of 0.62 nM.

Catalog NO:	CT-BZ001
Synonym:	Velcade
CAS NO:	179324-69-7
Mol. Formula:	C₁₉H₂₅BN₄O₄
MW:	384.24

** >99% pure, snow-white powder (pic attached), with clean and impeccable NMR. In stock. Prompt.

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NO	Size	Price	In Stock	Quantity
1	5 mg	$100.00	YES
2	25 mg	$380.00	YES

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Solubility : Soluble in DMSO, Methanol

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99% (HPLC)

Original QC Data : ¹H-NMR, HPLC and MS

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Bortezomib, Lot BZ-AE,Visual Appearance.pdf
Bortezomib, Lot BZ-AE, Certificate of Analysis.pdf

1. J. Adams, et al, Cancer Invest (2004) 22 (2), 304; J. Adams, et al, Bioorg. Med. Chem. Lett. (1998) 8, 333-338.

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