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Home > Kinase Inhibitors > IGF-1R > BMS-754807

BMS-754807

A potent, selective orally active antagonist of the insulin-like growth factor-1 receptor (IGF-1R)

Catalog NO:	CT-BMS75
Synonym:
CAS NO:	1001350-96-4
Mol. Formula:	C₂₃H₂₄FN₉O ∙ 1.6H₂O
MW:	490.3

** in vivo Quality Material. A clean, optically pure product. Dihydrate, validated by a spot-on Quantitative Elemental Analysis. Same Day Shipping.

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NO	Size	Price	In Stock	Quantity
1	5 mg	$100.00	YES
2	10 mg	$150.00	YES
3	50 mg	$400.00	YES
4	100 mg	$650.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : >99.5% Chem and optical purity (HPLC and Chiral HPLC)

Original QC Data : HPLC-MS, ¹HNMR, Chiral HPLC, and Quantitative Elemental Analysis

Please Pick Batch NO:

BMS-754807, Lot 03, 2xH2O, Certificate of Analysis.pdf

1. Witterman, M. D., et al, Discovery of a 2,4-Disubstituted Pyrrolo-[1,2-f][1,2,4]triazine Inhibitor (BMS-754807) of Insulin-like Growth Factor Receptor (IGF-1R) Kinase in Clinical Development, J. Med. Chem. published Sept 25, 2009

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