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Home > Kinase Inhibitors > mTOR > AZD8055

AZD8055

AZD8055 is a potent, orally bioavailable and ATP-competitive mTORC1/C2 inhibitor with an IC50 of 0.8 nM, highly selective ( ~1000 fold) over all class I PI3K isoforms and other PI3K-like kinase family, and there is no significant activity against a panel of other 260 kinases at a concentration up to 10,000 nM.

Catalog NO:	CT-A8055
Synonym:
CAS NO:	1009298-09-2
Mol. Formula:	C₂₅H₃₁N₅O₄
MW:	465.5

** Grams in stock from Indianapolis USA. A yellow solid/powder coming with an excellent Quantitative Elemental Analysis. Ship within 1 day

Pricing and OrderingTechnical Data

QC & Certificates

References

NO	Size	Price	In Stock	Quantity
1	10 mg	$60.00	YES
2	50 mg	$140.00	YES
3	100 mg	$227.00	YES
4	200 mg	$399.00	YES

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Solubility : Soluble in DMSO

Storage : Store at 0°C (short term), -20°C (long term), desiccated

Purity : 99% (HPLC at 214 and 254 nm)

Original QC Data : HPLC-MS, ¹HNMR, and Quantitative Elemental Analysis

Please Pick Batch NO:

AZD8055, Current Lot, Certificate of Analysis

1. C. M. Chresta, et al, AZD8055 Is a Potent, Selective, and Orally Bioavailable ATP-Competitive Mammalian Target of Rapamycin Kinase Inhibitor with In vitro and In vivo Antitumor Activity, Cancer Res. 2010, 70: 288-298.

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